Pinacidil potentiates morphine analgesia

Life Sci. 1992;50(16):PL135-8. doi: 10.1016/0024-3205(92)90467-4.

Abstract

The opening of K+ channels in the membrane of target neurons is a key mechanism of the effect of opioids. Here we show that the K+ channel opener, pinacidil, i.c.v. injected at doses of 50, 100 or 150 micrograms/rat, significantly increases and prolongs the effect of morphine on the thermal pain threshold (hot-plate and tail-flick tests). These data may suggest a novel approach to the management of pain.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Analgesia*
  • Animals
  • Dose-Response Relationship, Drug
  • Drug Synergism
  • Guanidines / administration & dosage*
  • Ion Channel Gating / drug effects
  • Male
  • Morphine / administration & dosage*
  • Pain / physiopathology
  • Pinacidil
  • Potassium Channels / drug effects
  • Rats
  • Rats, Inbred Strains

Substances

  • Guanidines
  • Potassium Channels
  • Morphine
  • Pinacidil