A selective, cell-permeable optical probe for hydrogen peroxide in living cells

J Am Chem Soc. 2004 Dec 1;126(47):15392-3. doi: 10.1021/ja0441716.

Abstract

We present the synthesis, properties, and biological applications of Peroxyfluor-1 (PF1), a new type of optical probe for intracellular imaging of hydrogen peroxide in living biological samples. PF1 utilizes a boronate deprotection mechanism to provide unprecedented selectivity and optical dynamic range for detecting H2O2 in aqueous solution over similar reactive oxygen species including superoxide, nitric oxide, tert-butyl hydroperoxide, and hydroxyl radical. We further demonstrate the value of this reagent for biological applications by imaging changes in [H2O2] in living mammalian cells.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Boronic Acids / chemistry
  • Cell Line
  • Cell Membrane Permeability
  • Esters / chemistry
  • Fluoresceins / chemical synthesis
  • Fluoresceins / chemistry*
  • Fluoresceins / metabolism
  • Fluoresceins / pharmacokinetics
  • Humans
  • Hydrogen Peroxide / analysis*
  • Microscopy, Confocal / methods
  • Microscopy, Fluorescence / methods
  • Substrate Specificity
  • Xanthenes / chemistry

Substances

  • Boronic Acids
  • Esters
  • Fluoresceins
  • Xanthenes
  • peroxyfluor-1
  • Hydrogen Peroxide