The anorectic effect of neurotensin is mediated via a histamine H1 receptor in mice

Peptides. 2004 Dec;25(12):2135-8. doi: 10.1016/j.peptides.2004.07.009.

Abstract

Neurotensin (NT), a tridecapeptide found in the mammalian brain and peripheral tissues, induces a decrease in food intake after central administration. In this investigation, we examine whether the histaminergic system is involved in NT-induced suppression of feeding. Intracerebroventricular injection of NT (0.1-1 nmol/mouse) led to dose-dependent inhibition of food intake in fasted ddY mice. The anorectic effect induced by NT (0.1 nmol/mouse) was ameliorated upon co-administration of pyrilamine (3 nmol/mouse), an antagonist for histomine H1 receptor. The NT-induced anorectic effect was partially ameliorated in H1 knockout mice. The findings suggest that the H1 receptor in part mediates the NT-induced suppression of food intake.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Appetite Depressants / pharmacology*
  • Eating / drug effects
  • Injections, Intraventricular
  • Male
  • Mice
  • Mice, Knockout
  • Neurotensin / physiology*
  • Receptors, Histamine H1 / physiology*

Substances

  • Appetite Depressants
  • Receptors, Histamine H1
  • Neurotensin