[Study on in vitro and in vivo antibacterial activity of pheromonicin-SA]

Sichuan Da Xue Xue Bao Yi Xue Ban. 2004 Nov;35(6):749-52.
[Article in Chinese]

Abstract

Objective: To evaluate the bactericidal activity of pheromonicin-SA (Ph-SA) via routine in vitro/in vivo measurement.

Methods: Minimal inhibitory concentration (MIC50 and MIC90) of Ph-SA were evaluated via in vitro double-dilution assay with 69 strains pathogenic bacteria and via intraperitoneal infected mice with intravenous Ph-SA treatment.

Results: In vitro data showed that bactericidal activity of Ph-SA was approximately 12 times greater, on a molar basis, than that of vancomycin. In vivo data showed that bactericidal activity of Ph-SA was approximately 59 times greater than that of vancomycin.

Conclusion: The results suggest that Ph-SA may be of potential value as antibiotic against methicillin-resistant Staphylococcus aureus (MRSA).

Publication types

  • English Abstract
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Anti-Bacterial Agents / pharmacology*
  • Bacterial Proteins / genetics*
  • Drug Resistance, Microbial
  • Female
  • Male
  • Methicillin Resistance
  • Mice
  • Microbial Sensitivity Tests
  • Peptide Biosynthesis
  • Peptides / genetics*
  • Peptides, Cyclic
  • Recombinant Fusion Proteins / biosynthesis
  • Recombinant Fusion Proteins / pharmacology
  • Staphylococcal Infections / drug therapy
  • Staphylococcus aureus / drug effects*
  • Vancomycin / pharmacology
  • Vancomycin / therapeutic use

Substances

  • AgrD protein, Staphylococcus
  • Anti-Bacterial Agents
  • Bacterial Proteins
  • Peptides
  • Peptides, Cyclic
  • Recombinant Fusion Proteins
  • Vancomycin