Spontaneous formation of nucleic acid-based nanoparticles is responsible for high interferon-alpha induction by CpG-A in plasmacytoid dendritic cells

J Biol Chem. 2005 Mar 4;280(9):8086-93. doi: 10.1074/jbc.M410868200. Epub 2004 Dec 8.

Abstract

Plasmacytoid dendritic cells (PDC) represent a highly specialized immune cell subset that produces large quantities of the anti-viral cytokines type I interferons (IFN-alpha and IFN-beta) upon viral infection. PDC employ a member of the family of toll-like receptors, TLR9, to detect CpG motifs (unmethylated CG dinucleotides in certain base context) present in viral DNA. A certain group of CpG motif-containing oligodeoxynucleotides (CpG ODN), CpG-A, was the first synthetic stimulus available that induced large amounts of interferon-alpha (IFN-alpha) in PDC. However, the mechanism responsible for this activity remained elusive. CpG-A is characterized by a central palindrome and poly(G) at the 5' and 3' end. Here we demonstrate that CpG-A self-assembles to higher order tertiary structures via G-tetrad formation of their poly(G) motifs. Spontaneous G-tetrad formation of CpG-A required the palindrome sequence allowing structure formation in a physiological environment. Once formed, G-tetrad-linked structures were stable even under denaturing conditions. Atomic force microscopy revealed that the tertiary structures formed by CpG-A represent nucleic acid-based nanoparticles in the size range of viruses. Similarly sized preformed polystyrene nanoparticles loaded with a CpG ODN that is otherwise weak at inducing IFN-alpha (CpG-B) gained the potency of CpG-A to induce IFN-alpha. Higher ODN uptake in PDC was not responsible for the higher IFN-alpha-inducing activity of CpG-A or of CpG-B-coated nanoparticles as compared with CpG-B. Based on these results we propose a model in which the spatial configuration of CpG motifs as particle is responsible for the virus-like potency of CpG-A to induce IFN-alpha in PDC.

MeSH terms

  • Adolescent
  • Adult
  • Aged
  • Buffers
  • Cells, Cultured
  • CpG Islands*
  • Cytokines / metabolism
  • DNA / chemistry
  • Dendritic Cells / cytology*
  • Electrophoresis, Polyacrylamide Gel
  • Flow Cytometry
  • Humans
  • Interferon-alpha / metabolism
  • Microscopy, Atomic Force
  • Middle Aged
  • Models, Genetic
  • Nanostructures / ultrastructure*
  • Nucleic Acid Conformation
  • Nucleic Acids / chemistry*
  • Oligonucleotides / chemistry
  • Plasma Cells / metabolism*
  • Polystyrenes / chemistry
  • Temperature

Substances

  • Buffers
  • Cytokines
  • Interferon-alpha
  • Nucleic Acids
  • Oligonucleotides
  • Polystyrenes
  • DNA