Effects of 15-deoxy-delta12,14-prostaglandin J2 on the cyclooxygenase-2 expression in the murine lung in the presence of lipopolysaccharide

Arzneimittelforschung. 2004;54(11):711-4. doi: 10.1055/s-0031-1297028.

Abstract

A previous study has demonstrated that 15-deoxy-delta12,14-prostaglandin J2 (15d-PG J2) enhanced acute lung injury induced by lipopolysaccharide (LPS) in mice. The enhancement in acute lung injury by 15d-PG J2 was concomitant with the enhanced expression of interleukin-1beta and chemokines in the lung. However, other underlying mechanisms of this enhancement remain to be elucidated. Cyclooxygenase (COX)-2 has been reported to be involved in enhanced pulmonary permeability during acute lung injury. This study investigated the effects of 15d-PG J2 on COXs expressions in the lung in the presence or absence of LPS. ICR mice were divided into 4 experimental groups that intratracheally received vehicle, lipopolysaccharide (LPS: 125 microg/kg), 15d-PG J2 (1 mg/kg), or 15d-PG J2 + LPS. The expression of mRNA for both COX-1 and -2 in the lung was evaluated 4 h after the intratracheal administration. 15d-PG J2 enhanced the COX-2 mRNA expression in the presence of LPS. In contrast, 15d-PG J2 did not affect the COX-1 expression. These results suggest that the enhancing effects of 15d-PG J2 on LPS-induced acute lung injury might be explained, at least in part, by those on the lung expression of COX-2.

MeSH terms

  • Animals
  • Bacterial Toxins / toxicity
  • Cyclooxygenase 1
  • Cyclooxygenase 2
  • Enterotoxins / toxicity
  • Escherichia coli Proteins / toxicity
  • Isoenzymes / biosynthesis*
  • Isoenzymes / genetics
  • Lipopolysaccharides / pharmacology
  • Lung / drug effects
  • Lung / enzymology*
  • Lung / pathology
  • Lung Diseases / chemically induced
  • Lung Diseases / enzymology
  • Lung Diseases / pathology
  • Male
  • Membrane Proteins
  • Mice
  • Mice, Inbred ICR
  • Prostaglandin D2 / analogs & derivatives*
  • Prostaglandin D2 / pharmacology*
  • Prostaglandin-Endoperoxide Synthases / biosynthesis*
  • Prostaglandin-Endoperoxide Synthases / genetics
  • RNA, Messenger / biosynthesis
  • Reverse Transcriptase Polymerase Chain Reaction

Substances

  • 15-deoxyprostaglandin J2
  • Bacterial Toxins
  • Enterotoxins
  • Escherichia coli Proteins
  • Isoenzymes
  • Lipopolysaccharides
  • Membrane Proteins
  • RNA, Messenger
  • heat-labile enterotoxin, E coli
  • Cyclooxygenase 1
  • Cyclooxygenase 2
  • Prostaglandin-Endoperoxide Synthases
  • Ptgs1 protein, mouse
  • Prostaglandin D2