Musk xylene is a novel specific inducer of cytochrome P-450IA2

Biochem Biophys Res Commun. 1992 Apr 15;184(1):149-53. doi: 10.1016/0006-291x(92)91171-l.

Abstract

The effect of musk xylene on contents of both cytochrome P-450IA1 and cytochrome P-450IA2 in rat liver was investigated using Western blotting analysis. Rats were treated i.p. for five consecutive days with either 50, 100 or 200 mg musk xylene/kg body weight. Musk xylene increased both total cytochrome P-450 and cytochrome b5 contents in rat liver microsomes. Musk xylene induced cytochrome P-450IA2 (384 pmol/mg protein) strongly and preferentially and the ratio of cytochrome P450IA2/P-450IA1 was about 12 at the lowest dose tested. Musk xylene also induced the cytochrome P-450IA1 dose-dependently, but these extents were very small (32-174 pmol/mg protein). These results suggest that musk xylene may be a more specific inducer for cytochrome P-450IA2 than any other inducers reported.

MeSH terms

  • Animals
  • Blotting, Western
  • Cytochrome P-450 CYP1A2
  • Cytochrome P-450 Enzyme System / biosynthesis*
  • Cytochromes b5 / biosynthesis
  • Dose-Response Relationship, Drug
  • Enzyme Induction
  • Kinetics
  • Male
  • Microsomes, Liver / drug effects
  • Microsomes, Liver / metabolism*
  • Oxidoreductases / biosynthesis*
  • Perfume
  • Rats
  • Rats, Inbred Strains
  • Reference Values
  • Xylenes / pharmacology*

Substances

  • Perfume
  • Xylenes
  • musk xylene
  • Cytochromes b5
  • Cytochrome P-450 Enzyme System
  • Oxidoreductases
  • Cytochrome P-450 CYP1A2