Characterization of the interaction between interleukin-13 and interleukin-13 receptors

J Biol Chem. 2005 Jul 1;280(26):24915-22. doi: 10.1074/jbc.M502571200. Epub 2005 May 3.

Abstract

Interleukin-13 (IL-13) possesses two types of receptor: the heterodimer, composed of the IL-13Ralpha1 chain (IL-13Ralpha1) and the IL-4Ralpha chain (IL-4Ralpha), transducing the IL-13 signals; and the IL-13Ralpha2 chain (IL-13Ralpha2), acting as a nonsignaling "decoy" receptor. Extracellular portions of both IL-13Ralpha1 and IL-13Ralpha2 are composed of three fibronectin type III domains, D1, D2, and D3, of which the last two comprise the cytokine receptor homology modules (CRHs), a common structure of the class I cytokine receptor superfamily. Thus far, there has been no information about the critical amino acids of the CRHs or the role of the D1 domains of IL-13Ralpha1 and IL-13Ralpha2 in binding to IL-13. In this study, we first built the homology modeling of the IL-13.hIL-13 receptor complexes and then predicted the amino acids involved in binding to IL-13. By incorporating mutations into these amino acids, we identified Tyr-207, Asp-271, Tyr-315, and Asp-318 in the CRH of human IL-13Ralpha2, and Leu-319 and Tyr-321 in the CRH of human IL-13Ralpha1, as critical residues for binding to IL-13. Tyr-315 in IL-13Ralpha2 and Leu-319 in IL-13Ralpha1 are positionally conserved hydrophobic amino acid residues. Furthermore, by using D1 domain-deleted mutants, we found that the D1 domain is needed for the expression of IL-13Ralpha2, but not IL-13Ralpha1, and that the D1 domain of IL-13Ralpha1 is important for binding to IL-13, but not to IL-4. These results provide the basis for a precise understanding of the interaction between IL-13 and its receptors.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Amino Acid Sequence
  • Binding Sites
  • Cytokines / metabolism
  • Dimerization
  • Dose-Response Relationship, Drug
  • Fibronectins / chemistry
  • Gene Deletion
  • Humans
  • Interleukin-13 / chemistry*
  • Interleukin-13 Receptor alpha1 Subunit
  • Interleukin-4 / metabolism
  • Kinetics
  • Luciferases / metabolism
  • Models, Biological
  • Models, Genetic
  • Models, Molecular
  • Molecular Sequence Data
  • Mutagenesis
  • Mutation
  • Protein Binding
  • Protein Structure, Tertiary
  • Receptors, Interleukin / chemistry*
  • Receptors, Interleukin-13
  • Recombinant Proteins / chemistry
  • Sequence Homology, Amino Acid
  • Signal Transduction

Substances

  • Cytokines
  • Fibronectins
  • IL13RA1 protein, human
  • Interleukin-13
  • Interleukin-13 Receptor alpha1 Subunit
  • Receptors, Interleukin
  • Receptors, Interleukin-13
  • Recombinant Proteins
  • Interleukin-4
  • Luciferases