Effects of inducible overexpression of DNp73alpha on cancer cell growth and response to treatment in vitro and in vivo

Cell Death Differ. 2005 Jul;12(7):805-14. doi: 10.1038/sj.cdd.4401622.

Abstract

The p73 gene has a complex regulation, which leads to the expression of different isoforms, often with opposite biological effects. We have generated in the human colocarcinoma cell line HCT116, expressing a wild-type p53, an inducible DNp73alpha expressing system. Two clones (HCT116/DN3 and HCT116/DN14), upon doxycycline addition, show a strong expression of DNp73alpha. In vitro the two DNp73alpha overexpressing clones grow at similar rate of the control transfected clone (HCT116/8a) and similarly respond to DNA damage. When injected in mice, HCT116/DN3, HCT116/DN14, and HCT116/8a cells grew similarly in the absence or presence of tetracycline. In HCT116/DN3 and HCT116/DN14 tumors, tetracycline induced a strong expression of DNp73alpha both as mRNA and protein. These results indicate that in this system the overexpression of the DNp73alpha does not induce a more aggressive phenotype and does not seem to be associated with a reduced response of the cells to treatment with anticancer agents.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Antibiotics, Antineoplastic / pharmacology
  • Cell Proliferation / drug effects
  • DNA Damage / drug effects
  • DNA-Binding Proteins / genetics*
  • DNA-Binding Proteins / metabolism*
  • Doxorubicin / pharmacology
  • Doxycycline / pharmacology
  • Gene Expression
  • Genes, Tumor Suppressor
  • HCT116 Cells
  • Humans
  • Mice
  • Neoplasms / drug therapy*
  • Neoplasms / genetics
  • Neoplasms / pathology*
  • Nuclear Proteins / genetics*
  • Nuclear Proteins / metabolism*
  • Phenotype
  • Tumor Protein p73
  • Tumor Suppressor Proteins

Substances

  • Antibiotics, Antineoplastic
  • DNA-Binding Proteins
  • Nuclear Proteins
  • TP73 protein, human
  • Trp73 protein, mouse
  • Tumor Protein p73
  • Tumor Suppressor Proteins
  • Doxorubicin
  • Doxycycline