7-day rescue therapy with ranitidine bismuth citrate after Helicobacter pylori treatment failure

Aliment Pharmacol Ther. 2005 May 15;21(10):1249-53. doi: 10.1111/j.1365-2036.2005.02465.x.

Abstract

Background: Quadruple rescue therapy requires a complex scheme with four drugs.

Aim: To evaluate the efficacy of ranitidine bismuth citrate-tetracycline-metronidazole rescue regimen, and to compare two different metronidazole dose schemes.

Methods: Prospective multicentre study including proton-pump inhibitor + clarithromycin + amoxicillin failures. Rescue regimen included two 7-day treatment: (i) ranitidine bismuth citrate (400 mg b.d.)-tetracycline (500 mg q.d.s.)-metronidazole (500 mg t.d.s.; RTM1); or (ii) the same regimen but with metronidazole 250 mg q.d.s. (RTM2). Eradication was confirmed with (13)C-urea breath test.

Results: A total of 150 patients were included (58 RTM1, 92 RTM2). All patients but two (one in each group) returned after treatment. About 86% in group RTM1 and 95% in RTM2 correctly took all the medications (P = 0.076). Per-protocol eradication rates with RTM1 and RTM2 were 74 (95% CI: 60-84) and 69% (59-78). The intention-to-treat eradication rates were 64 (51-75) and 70% (59-78; P > 0.05). The type of regimen was not associated with eradication in the multivariate analysis. Adverse effects were more frequent with RTM1 (41%) than with RTM2 (30%; P > 0.05).

Conclusion: Seven-day triple rescue therapy with ranitidine bismuth citrate-tetracycline-metronidazole is effective for Helicobacter pylori eradication, and represents an encouraging alternative to quadruple therapy, with the advantage of simplicity. The administration of metronidazole every 6 h (together with tetracycline), and at a low dose (250 mg), achieves similar efficacy and is probably associated with a better compliance and a lower incidence of adverse effects.

Publication types

  • Clinical Trial
  • Comparative Study
  • Multicenter Study
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adult
  • Anti-Ulcer Agents / therapeutic use*
  • Bismuth / therapeutic use*
  • Dose-Response Relationship, Drug
  • Drug Combinations
  • Drug Therapy, Combination / therapeutic use
  • Female
  • Helicobacter Infections / drug therapy*
  • Helicobacter pylori*
  • Histamine H2 Antagonists / therapeutic use*
  • Humans
  • Male
  • Metronidazole / administration & dosage
  • Metronidazole / therapeutic use
  • Middle Aged
  • Prospective Studies
  • Ranitidine / analogs & derivatives*
  • Ranitidine / therapeutic use*
  • Tetracycline / therapeutic use
  • Treatment Failure

Substances

  • Anti-Ulcer Agents
  • Drug Combinations
  • Histamine H2 Antagonists
  • Metronidazole
  • ranitidine bismuth citrate
  • Ranitidine
  • Tetracycline
  • Bismuth