Fibrillin-1 interactions with heparin. Implications for microfibril and elastic fiber assembly

J Biol Chem. 2005 Aug 26;280(34):30526-37. doi: 10.1074/jbc.M501390200. Epub 2005 Jun 24.

Abstract

Fibrillin-1 assembly into microfibrils and elastic fiber formation involves interactions with glycosaminoglycans. We have used BIAcore technology to investigate fibrillin-1 interactions with heparin and with heparin saccharides that are analogous to S-domains of heparan sulfate. We have identified four high affinity heparin-binding sites on fibrillin-1, localized three of these sites, and defined their binding kinetics. Heparin binding to the fibrillin-1 N terminus has particularly rapid kinetics. Hyaluronan and chondroitin sulfate did not interact significantly with fibrillin-1. Heparin saccharides with more than 12 monosaccharide units bound strongly to all four fibrillin-1 sites. Heparin did not inhibit fibrillin-1 N- and C-terminal interactions or RGD-dependent cell attachment, but heparin and MAGP-1 competed for binding to the fibrillin-1 N terminus, and heparin and tropoelastin competed for binding to a central fibrillin-1 sequence. By regulating these key interactions, heparin can profoundly influence microfibril and elastic fiber assembly.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Biotin / chemistry
  • Biotinylation
  • Calcium / metabolism
  • Carbohydrate Sequence
  • Contractile Proteins / chemistry
  • Databases, Protein
  • Edetic Acid / chemistry
  • Exons
  • Extracellular Matrix Proteins / chemistry
  • Fibrillin-1
  • Fibrillins
  • Glycosaminoglycans / chemistry
  • Glycosylation
  • Heparin / chemistry*
  • Heparitin Sulfate / chemistry
  • Humans
  • Kinetics
  • Microfilament Proteins / chemistry*
  • Microfilament Proteins / metabolism
  • Models, Chemical
  • Models, Molecular
  • Molecular Sequence Data
  • Monosaccharides / chemistry
  • Oligosaccharides / chemistry
  • Protein Binding
  • Protein Structure, Tertiary
  • RNA Splicing Factors
  • Recombinant Proteins / chemistry
  • Swine
  • Time Factors
  • Tropoelastin / chemistry

Substances

  • Contractile Proteins
  • Extracellular Matrix Proteins
  • FBN1 protein, human
  • Fibrillin-1
  • Fibrillins
  • Glycosaminoglycans
  • Microfilament Proteins
  • Monosaccharides
  • Oligosaccharides
  • RNA Splicing Factors
  • Recombinant Proteins
  • Tropoelastin
  • microfibrillar protein
  • Biotin
  • Heparin
  • Heparitin Sulfate
  • Edetic Acid
  • Calcium