First aldehyde-functionalized poly(2-oxazoline)s for chemoselective ligation

Macromol Biosci. 2005 Jul 14;5(7):603-12. doi: 10.1002/mabi.200500059.

Abstract

A protected aldehyde-functionalized 2-oxazoline, 2-[3-(1,3)-dioxolan-2-ylpropyl]-2-oxazoline (DPOx), was synthesized from commercially available compounds in high yields. The polymerization of DPOx with different initiators proceeds via a living ionic mechanism; thus, the polymers were of low polydispersity and the degree of polymerization could be precisely adjusted. Copolymerization with 2-methyl-2-oxazoline gave water-soluble statistical copolymers. Hydrolysis of the homo- and copolymers resulted in well-defined, aldehyde-bearing poly(2-oxazoline)s. The aldehyde side functions reacted quantitatively with an amino-oxy compound to form the corresponding oxime.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Aldehydes / chemistry*
  • Dioxolanes / chemical synthesis*
  • Oxazoles / chemical synthesis*
  • Polymers / chemical synthesis*

Substances

  • 2-(3-(1,3)-dioxolan-2-ylpropyl)-2-oxazoline
  • Aldehydes
  • Dioxolanes
  • Oxazoles
  • Polymers