A new point-of-care method for monitoring anti-platelet therapy: application of the cone and plate(let) analyzer

Platelets. 2005 Aug;16(5):293-9. doi: 10.1080/09537100400028800.

Abstract

Recent studies suggest that anti-platelet agents are not equally effective in all individuals. We have developed a new method to evaluate the effect of anti-platelet drugs using the cone and plate(let) analyzer (CPA) test. The method is based on the ability of activators to reduce platelet adhesion under flow conditions. Treatment of a blood sample with arachidonic acid (AA) or ADP in vitro significantly decreased platelet deposition to a surface coverage (SC) of 2.1+/-0.4 and 1.3+/-0.6%, respectively, compared with the basic SC of 12.3+/-6.8%. The effect of AA was prevented by aspirin (SC 8.1+/-3.8%) and that of ADP was reduced by 2-methylthio-AMP, a P2Y12 ADP receptor inhibitor (SC 4.8+/-2.0%). Pre-incubation with AA of whole blood samples from untreated healthy volunteers resulted in a marked decline of SC (from SC 9.8+/-2.2 to 0.6+/-0.3%). In contrast, in volunteers treated with 100, 300, and 500 mg aspirin per day, AA (but not ADP) decreased SC only to 3.5+/-1.3, 4.4+/-1.7, and 4.1+/-2.0%, respectively (P<0.001 versus SC with AA before treatment). A good correlation was observed between the modified CPA and aggregometry (R2=0.55). In conclusion, the modified CPA test is a useful tool to evaluate the efficacy of anti-platelet therapy.

MeSH terms

  • Adenosine Diphosphate / pharmacology
  • Adult
  • Arachidonic Acid / pharmacology
  • Aspirin / blood
  • Aspirin / pharmacology
  • Blood Proteins / pharmacology
  • Drug Monitoring / methods*
  • Humans
  • Membrane Proteins / antagonists & inhibitors
  • Membrane Proteins / blood
  • Membrane Proteins / pharmacology
  • Platelet Adhesiveness / drug effects
  • Platelet Aggregation Inhibitors / pharmacology*
  • Platelet Function Tests / instrumentation
  • Platelet Function Tests / methods*
  • Point-of-Care Systems*
  • Purinergic P2 Receptor Antagonists
  • Receptors, Purinergic P2 / blood
  • Receptors, Purinergic P2Y12
  • Sensitivity and Specificity

Substances

  • Blood Proteins
  • Membrane Proteins
  • P2RY12 protein, human
  • Platelet Aggregation Inhibitors
  • Purinergic P2 Receptor Antagonists
  • Receptors, Purinergic P2
  • Receptors, Purinergic P2Y12
  • platelet adhesion inhibitor
  • Arachidonic Acid
  • Adenosine Diphosphate
  • Aspirin