Sustained vascular endothelial growth factor delivery enhances angiogenesis and perfusion in ischemic hind limb

Pharm Res. 2005 Jul;22(7):1110-6. doi: 10.1007/s11095-005-5644-2. Epub 2005 Jul 22.

Abstract

Purpose: We hypothesized that sustained delivery of vascular endothelial growth factor (VEGF) using a polymer [85:15 poly(lactide-co-glycolide) (PLG)] would enhance angiogenesis and improve perfusion of ischemic tissue.

Methods: C57BL/6J mice (n = 20/group) underwent unilateral hind limb ischemia surgery and were randomized to groups of no scaffold implantation (0-Implant), unloaded scaffold implantation (Empty-PLG), or implantation of scaffolds incorporating 3 microg of VEGF165 (PLG-VEGF). Endpoints included laser Doppler perfusion imaging (LDPI, ischemic/nonischemic limb, %), local vessel counts, immunohistochemistry for CD31, and alpha-smooth muscle actin. In vitro release kinetics of VEGF from PLG was also measured.

Results: PLG-VEGF resulted in improved lower extremity perfusion vs. controls as measured by LDPI% at 7, 14, 21, and 28 days (p < 0.05). PLG-VEGF was associated with significantly greater percentage of vessels staining for CD31 and alpha-smooth muscle actin compared to the Empty-PLG or 0-Implant (p < 0.05 for both).

Conclusions: The PLG-VEGF scaffolds resulted in sustained VEGF delivery, improved tissue perfusion, greater capillary density, and more mature vasculature compared to the controls. The sustained-release PLG polymer vehicle is a promising delivery system for therapeutic neovascularization applications.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • Actins / metabolism
  • Animals
  • Biocompatible Materials / administration & dosage
  • Capillaries / growth & development
  • Disease Models, Animal
  • Drug Carriers
  • Hindlimb / blood supply
  • Hindlimb / physiopathology
  • Humans
  • Ischemia / drug therapy*
  • Ischemia / physiopathology
  • Lactic Acid / administration & dosage*
  • Laser-Doppler Flowmetry
  • Male
  • Mice
  • Mice, Inbred C57BL
  • Muscle, Skeletal / blood supply*
  • Muscle, Skeletal / physiopathology
  • Neovascularization, Physiologic* / drug effects
  • Perfusion
  • Platelet Endothelial Cell Adhesion Molecule-1 / metabolism
  • Polyglycolic Acid / administration & dosage*
  • Polylactic Acid-Polyglycolic Acid Copolymer
  • Polymers / administration & dosage*
  • Vascular Endothelial Growth Factor A / administration & dosage*

Substances

  • Actins
  • Biocompatible Materials
  • Drug Carriers
  • Platelet Endothelial Cell Adhesion Molecule-1
  • Polymers
  • Vascular Endothelial Growth Factor A
  • Polylactic Acid-Polyglycolic Acid Copolymer
  • Polyglycolic Acid
  • Lactic Acid