Bcr-Abl activates the AKT/Fox O3 signalling pathway to restrict transforming growth factor-beta-mediated cytostatic signals

EMBO Rep. 2005 Oct;6(10):985-91. doi: 10.1038/sj.embor.7400501.

Abstract

The fusion of Abl with either Bcr or Tel in human leukaemia leads to the constitutive activation of Abl tyrosine kinase, which in turn induces growth-factor-independent proliferation and cell survival. However, the mechanism by which Bcr-Abl induces cellular transformation has not yet been well characterized. Here, we show that Bcr-Abl-expressing cells are resistant to growth inhibition and apoptosis mediated by transforming growth factor-beta (TGF-beta). Interestingly, we observed that the suppressive effects of Bcr-Abl on TGF-beta responses were not mediated by an impairment of Smad signalling, which is believed to act as the principal mediator of TGF-beta responses. In contrast, we found that Bcr-Abl can target the protein kinase AKT and the transcription factor Fox O3 to interfere with growth inhibition and apoptosis in response to TGF-beta. Our results show a novel mechanism of cellular transformation by the oncogenic fusion protein Bcr-Abl through suppression of the cytostatic actions of TGF-beta.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Apoptosis
  • Blotting, Western
  • Cell Line
  • Cell Proliferation
  • Fluorescent Antibody Technique
  • Forkhead Transcription Factors / physiology*
  • Fusion Proteins, bcr-abl / physiology*
  • Humans
  • Mice
  • Phosphatidylinositol 3-Kinases / physiology
  • Phosphorylation
  • Proto-Oncogene Proteins c-akt / physiology*
  • Signal Transduction / physiology*
  • Transforming Growth Factor beta / biosynthesis
  • Transforming Growth Factor beta / physiology*

Substances

  • Forkhead Transcription Factors
  • Transforming Growth Factor beta
  • Phosphatidylinositol 3-Kinases
  • Fusion Proteins, bcr-abl
  • Proto-Oncogene Proteins c-akt