Phase I/II combined chemoimmunotherapy with carcinoembryonic antigen-derived HLA-A2-restricted CAP-1 peptide and irinotecan, 5-fluorouracil, and leucovorin in patients with primary metastatic colorectal cancer

Clin Cancer Res. 2005 Aug 15;11(16):5993-6001. doi: 10.1158/1078-0432.CCR-05-0018.

Abstract

Purpose: We conducted a phase I/II randomized trial to evaluate the clinical and immunologic effect of chemotherapy combined with vaccination in primary metastatic colorectal cancer patients with a carcinoembryonic antigen-derived peptide in the setting of adjuvants granulocyte macrophage colony-stimulating factor, CpG-containing DNA molecules (dSLIM), and dendritic cells.

Experimental design: HLA-A2-positive patients with confirmed newly diagnosed metastatic colorectal cancer and elevated serum carcinoembryonic antigen (CEA) were randomized to receive three cycles of standard chemotherapy (irinotecan/high-dose 5-fluorouracil/leucovorin) and vaccinations with CEA-derived CAP-1 peptide admixed with different adjuvants [CAP-1/granulocyte macrophage colony-stimulating factor/interleukin-2 (IL-2), CAP-1/dSLIM/IL-2, and CAP-1/IL-2]. After completion of chemotherapy, patients received weekly vaccinations until progression of disease. Immune assessment was done at baseline and after three cycles of combined chemoimmunotherapy. HLA-A2 tetramers complexed with the peptides CAP-1, human T-cell lymphotrophic virus type I TAX, cytomegalovirus (CMV) pp65, and EBV BMLF-1 were used for phenotypic immune assessment. IFN-gamma intracellular cytokine assays were done to evaluate CTL reactivity.

Results: Seventeen metastatic patients were recruited, of whom 12 completed three cycles. Therapy resulted in five complete response, one partial response, five stable disease, and six progressive disease. Six grade 1 local skin reactions and one mild systemic reaction to vaccination treatment were observed. Overall survival after a median observation time of 29 months was 17 months with a survival rate of 35% (6 of 17) at that time. Eight patients (47%) showed elevation of CAP-1-specific CTLs. Neither of the adjuvants provided superiority in eliciting CAP-1-specific immune responses. During three cycles of chemotherapy, EBV/CMV recall antigen-specific CD8+ cells decreased by an average 14%.

Conclusions: The presented chemoimmunotherapy is a feasible and safe combination therapy with clinical and immunologic efficacy. Despite concurrent chemotherapy, increases in CAP-1-specific T cells were observed in 47% of patients after vaccination.

Publication types

  • Clinical Trial, Phase I
  • Clinical Trial, Phase II
  • Randomized Controlled Trial
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Adult
  • Aged
  • Antineoplastic Combined Chemotherapy Protocols / therapeutic use*
  • CD3 Complex / analysis
  • CD4 Antigens / analysis
  • CD8 Antigens / analysis
  • Camptothecin / administration & dosage
  • Camptothecin / analogs & derivatives
  • Carcinoembryonic Antigen / blood
  • Carcinoembryonic Antigen / immunology*
  • Colorectal Neoplasms / immunology
  • Colorectal Neoplasms / pathology
  • Colorectal Neoplasms / therapy*
  • Combined Modality Therapy
  • Dose-Response Relationship, Drug
  • Female
  • Flow Cytometry
  • Fluorouracil / administration & dosage
  • Granulocyte-Macrophage Colony-Stimulating Factor / administration & dosage
  • HLA-A2 Antigen / immunology*
  • Humans
  • Immunodominant Epitopes / immunology
  • Immunotherapy / methods
  • Interferon-gamma / metabolism
  • Interleukin-2 / administration & dosage
  • Irinotecan
  • Leucovorin / administration & dosage
  • Liver Neoplasms / immunology
  • Liver Neoplasms / secondary
  • Liver Neoplasms / therapy
  • Male
  • Middle Aged
  • Oligopeptides / administration & dosage
  • Oligopeptides / immunology
  • Oligopeptides / therapeutic use*
  • Prospective Studies
  • T-Lymphocytes / cytology
  • T-Lymphocytes / drug effects
  • T-Lymphocytes / immunology
  • Treatment Outcome

Substances

  • CD3 Complex
  • CD4 Antigens
  • CD8 Antigens
  • Carcinoembryonic Antigen
  • HLA-A2 Antigen
  • Immunodominant Epitopes
  • Interleukin-2
  • Oligopeptides
  • Irinotecan
  • Interferon-gamma
  • Granulocyte-Macrophage Colony-Stimulating Factor
  • Leucovorin
  • Fluorouracil
  • Camptothecin