Induction of a proinflammatory program in normal human thyrocytes by the RET/PTC1 oncogene

Proc Natl Acad Sci U S A. 2005 Oct 11;102(41):14825-30. doi: 10.1073/pnas.0503039102. Epub 2005 Oct 3.

Abstract

Rearrangements of the RET receptor tyrosine kinase gene generating RET/PTC oncogenes are specific to papillary thyroid carcinoma (PTC), the most frequent thyroid tumor. Here, we show that the RET/PTC1 oncogene, when exogenously expressed in primary normal human thyrocytes, induces the expression of a large set of genes involved in inflammation and tumor invasion, including those encoding chemokines (CCL2, CCL20, CXCL8, and CXCL12), chemokine receptors (CXCR4), cytokines (IL1B, CSF-1, GM-CSF, and G-CSF), matrix-degrading enzymes (metalloproteases and urokinase-type plasminogen activator and its receptor), and adhesion molecules (L-selectin). This effect is strictly dependent on the presence of the RET/PTC1 Tyr-451 (corresponding to RET Tyr-1062 multidocking site). Selected relevant genes (CCL20, CCL2, CXCL8, CXCR4, L-selectin, GM-CSF, IL1B, MMP9, UPA, and SPP1/OPN) were found up-regulated also in clinical samples of PTC, particularly those characterized by RET/PTC activation, local extrathyroid spread, and lymph node metastases, when compared with normal thyroid tissue or follicular thyroid carcinoma. These results, demonstrating that the RET/PTC1 oncogene activates a proinflammatory program, provide a direct link between a transforming human oncogene, inflammation, and malignant behavior.

Publication types

  • Comparative Study
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Blotting, Western
  • Cell Movement / physiology
  • Cells, Cultured
  • Cytokines / metabolism
  • Enzyme-Linked Immunosorbent Assay
  • Gene Expression Regulation / genetics*
  • Gene Rearrangement / genetics*
  • Humans
  • Inflammation / genetics
  • Inflammation / metabolism*
  • L-Selectin / metabolism
  • Metalloproteases / metabolism
  • Microarray Analysis
  • Polymerase Chain Reaction
  • Proto-Oncogene Proteins c-ret / genetics
  • Proto-Oncogene Proteins c-ret / metabolism*
  • Receptors, Cytokine / metabolism
  • Thyroid Gland / cytology
  • Thyroid Gland / metabolism*
  • Thyroid Neoplasms / genetics
  • Thyroid Neoplasms / metabolism*
  • Urokinase-Type Plasminogen Activator / metabolism

Substances

  • Cytokines
  • Receptors, Cytokine
  • L-Selectin
  • Proto-Oncogene Proteins c-ret
  • RET protein, human
  • Metalloproteases
  • Urokinase-Type Plasminogen Activator