ATP-induced apoptosis of thymocytes is mediated by activation of P2 X 7 receptor and involves de novo ceramide synthesis and mitochondria

Biochim Biophys Acta. 2006 Jan;1761(1):73-82. doi: 10.1016/j.bbalip.2005.10.001. Epub 2005 Oct 24.

Abstract

Thymocytes were reported to undergo apoptosis in the presence of extracellular ATP through the activation of the purinergic receptors P2 X 1R, P2 X 7R or both. We investigated the identity of the P2 X R and the signaling pathways involved in ATP-mediated apoptosis. Apoptosis elicited by ATP was prevented by inhibition of P2 X 7R, or in thymocytes bearing a mutated P2 X 7R, and reproduced with a P2 X 7R agonist, but not with a P2 X 1R agonist. Stimulation of thymocytes with either ATP or a P2 X 7R agonist was found to stimulate a late de novo ceramide synthesis and mitochondrial alterations. Inhibition of either processes attenuated apoptosis. Interestingly, stimulation with either ATP or a P2 X 1R agonist induced an early ceramide accumulation and a weak caspases-3/7 activation that did not lead to apoptosis. In conclusion, de novo ceramide generation and mitochondrial alterations, both resulting from P2 X 7R activation, were implicated in ATP-induced thymocyte apoptosis.

MeSH terms

  • Adenosine Triphosphate / pharmacology*
  • Animals
  • Apoptosis / drug effects
  • Apoptosis / physiology*
  • Cells, Cultured
  • Ceramides / metabolism*
  • Kinetics
  • Mice
  • Mice, Inbred BALB C
  • Mitochondria / drug effects
  • Mitochondria / physiology*
  • Purinergic P2 Receptor Agonists
  • Receptors, Purinergic P2 / drug effects
  • Receptors, Purinergic P2 / physiology*
  • Receptors, Purinergic P2X7
  • Sphingosine / metabolism
  • T-Lymphocytes / drug effects
  • T-Lymphocytes / physiology*

Substances

  • Ceramides
  • P2rx7 protein, mouse
  • Purinergic P2 Receptor Agonists
  • Receptors, Purinergic P2
  • Receptors, Purinergic P2X7
  • Adenosine Triphosphate
  • Sphingosine