Protease nexin-2/amyloid beta-protein precursor limits cerebral thrombosis

Proc Natl Acad Sci U S A. 2005 Dec 13;102(50):18135-40. doi: 10.1073/pnas.0507798102. Epub 2005 Dec 5.

Abstract

The amyloid beta-protein precursor (AbetaPP) is best known as the parent molecule to the amyloid beta-peptide that accumulates in the brains of patients with Alzheimer's disease. Secreted isoforms of AbetaPP that contain the Kunitz proteinase inhibitor domain are analogous to the previously identified cell-secreted proteinase inhibitor known as protease nexin-2 (PN2). Although PN2/AbetaPP is enriched in brain and in circulating blood platelets, little is understood of its physiological function and potential role in disease processes outside of amyloid beta-peptide generation. We hypothesized that the potent inhibition of certain procoagulant proteinases by PN2/AbetaPP, coupled with its abundance in platelets and brain, indicate that it may function to regulate cerebral thrombosis. Here we show that specific and modest 2-fold overexpression of PN2/AbetaPP in circulating platelets of transgenic mice caused a marked inhibition of thrombosis in vivo. In contrast, deletion of PN2/AbetaPP in AbetaPP gene knockout mice resulted in a significant increase in thrombosis. Similarly, platelet PN2/AbetaPP transgenic mice developed larger hematomas in experimental intracerebral hemorrhage, whereas AbetaPP gene knockout mice exhibited reduced hemorrhage size. These findings indicate that PN2/AbetaPP plays a significant role in regulating cerebral thrombosis and that modest increases in this protein can profoundly enhance cerebral hemorrhage.

Publication types

  • Comparative Study
  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Amyloid beta-Protein Precursor / genetics
  • Amyloid beta-Protein Precursor / metabolism*
  • Animals
  • Blood Platelets / metabolism
  • Brain / metabolism
  • DNA Primers
  • Gene Expression*
  • Immunoblotting
  • Intracranial Thrombosis / etiology
  • Intracranial Thrombosis / metabolism*
  • Intracranial Thrombosis / pathology
  • Mice
  • Mice, Knockout
  • Mice, Transgenic
  • Partial Thromboplastin Time
  • Platelet Activation / physiology
  • Protease Nexins
  • Receptors, Cell Surface / genetics
  • Receptors, Cell Surface / metabolism*

Substances

  • Amyloid beta-Protein Precursor
  • DNA Primers
  • Protease Nexins
  • Receptors, Cell Surface