The role of Ca2+ in (-)-menthol-induced human promyelocytic leukemia HL-60 cell death

In Vivo. 2006 Jan-Feb;20(1):69-75.

Abstract

A human promyelocytic leukemia HL-60 cell line was selected to examine the effect of (-)-Menthol on cell death. Based on the results from morphological changes and the percentage of viable cells in HL-60 cells after treatment with various concentrations of (-)-Menthol, it was shown that (-)-Menthol induced cell death through necrosis, not apoptosis. No cell cycle arrest was found in HL-60 cells examined by flow cytometry analysis. Also, the DNA gel electrophoresis method showed that (-)-Menthol did not induce apoptosis in HL-60 cells. However, it was found that (-)-Menthol induced the production of Ca2+ in these examined cells, dose-dependently. When HL-60 cells were pretreated with the chelator (BAPTA) of Ca2+ for 3 hours before addition of (-)-Menthol to the culture, a decrease of Ca2+ production was observed. Under the same conditions, the percentage of viable HL-60 cells was increased. Apparently Ca2+ production is associated with the induction of (-)-Menthol-induced cell death.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Acetylation
  • Calcium / physiology*
  • Cell Death / drug effects*
  • Cell Death / physiology*
  • DNA Fragmentation
  • Egtazic Acid / administration & dosage
  • Egtazic Acid / analogs & derivatives
  • Electrophoresis
  • Fluorenes / metabolism
  • HL-60 Cells
  • Humans
  • Leukemia, Promyelocytic, Acute / pathology*
  • Menthol / pharmacology*

Substances

  • Fluorenes
  • Menthol
  • 2-aminofluorene
  • Egtazic Acid
  • 1,2-bis(2-aminophenoxy)ethane-N,N,N',N'-tetraacetic acid
  • Calcium