HIF-2alpha regulates Oct-4: effects of hypoxia on stem cell function, embryonic development, and tumor growth

Genes Dev. 2006 Mar 1;20(5):557-70. doi: 10.1101/gad.1399906.

Abstract

The division, differentiation, and function of stem cells and multipotent progenitors are influenced by complex signals in the microenvironment, including oxygen availability. Using a genetic "knock-in" strategy, we demonstrate that targeted replacement of the oxygen-regulated transcription factor HIF-1alpha with HIF-2alpha results in expanded expression of HIF-2alpha-specific target genes including Oct-4, a transcription factor essential for maintaining stem cell pluripotency. We show that HIF-2alpha, but not HIF-1alpha, binds to the Oct-4 promoter and induces Oct-4 expression and transcriptional activity, thereby contributing to impaired development in homozygous Hif-2alpha KI/KI embryos, defective hematopoietic stem cell differentiation in embryoid bodies, and large embryonic stem cell (ES)-derived tumors characterized by altered cellular differentiation. Furthermore, loss of HIF-2alpha severely reduces the number of embryonic primordial germ cells, which require Oct-4 expression for survival and/or maintenance. These results identify Oct-4 as a HIF-2alpha-specific target gene and indicate that HIF-2alpha can regulate stem cell function and/or differentiation through activation of Oct-4, which in turn contributes to HIF-2alpha's tumor promoting activity.

Publication types

  • Comparative Study
  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Alleles
  • Animals
  • Basic Helix-Loop-Helix Transcription Factors / genetics
  • Basic Helix-Loop-Helix Transcription Factors / metabolism*
  • Cell Hypoxia / genetics
  • Cell Hypoxia / physiology*
  • Cell Transformation, Neoplastic
  • Down-Regulation
  • Embryonic Development / genetics
  • Embryonic Development / physiology*
  • Female
  • Immunohistochemistry
  • Mice
  • Mice, Nude
  • Models, Genetic
  • Octamer Transcription Factor-3 / genetics
  • Octamer Transcription Factor-3 / metabolism*
  • Pregnancy
  • RNA, Messenger / metabolism
  • Stem Cells / cytology
  • Stem Cells / metabolism
  • Stem Cells / physiology*
  • Teratoma / genetics
  • Teratoma / metabolism*
  • Teratoma / pathology
  • Transforming Growth Factor alpha / metabolism
  • Vascular Endothelial Growth Factor A / metabolism

Substances

  • Basic Helix-Loop-Helix Transcription Factors
  • Octamer Transcription Factor-3
  • RNA, Messenger
  • Transforming Growth Factor alpha
  • Vascular Endothelial Growth Factor A
  • endothelial PAS domain-containing protein 1