Synthesis and antiviral evaluation of novel open-chain analogues of neplanocin A

Nucleosides Nucleotides Nucleic Acids. 2006 Mar;25(3):341-50. doi: 10.1080/15257770500544578.

Abstract

Novel acyclic nucleoside analogues were designed and synthesized as open-chain analogues of neplanocin A. The coupling of the allylic bromide with purine bases using cesium carbonate afforded a series of novel acyclic nucleosides. The synthesized compounds Ia-II were evaluated for their antiviral activity against various viruses such as HIV HSV-1, HSV-2, and ECMV.

MeSH terms

  • Adenosine / analogs & derivatives*
  • Adenosine / chemical synthesis
  • Adenosine / pharmacology
  • Antiviral Agents / chemical synthesis*
  • Antiviral Agents / pharmacology*
  • Cell Line
  • Herpesvirus 1, Human / drug effects
  • Herpesvirus 2, Human / drug effects
  • Humans

Substances

  • Antiviral Agents
  • neplanocin A
  • Adenosine