Modulation of infectivity in phage display as a tool to determine the substrate specificity of proteases

Chembiochem. 2006 Jun;7(6):965-70. doi: 10.1002/cbic.200600051.

Abstract

Proteases play an important role in human and animal diseases. Rapid determination of substrate specificity is possible through the use of substrate phage display; however, current methods possess several drawbacks. They require phage-immobilization and cannot be used for infectivity-destroying or affinity tag-destroying proteases; this can make entire libraries useless. To overcome these limitations, here we introduce infectivity-modulated phage display (IMOP). IMOP uses a protease-resistant and infectivity-reducing tag fused to substrate-displaying polyvalent phages, and the specific cleavage of the substrate increases the infectivity of the phages by releasing the infectivity-reducing tag. The resulting phages were first tested with the infectivity-destroying detergent protease subtilisin; this resulted in a highly specific substrate at a 200-fold enrichment. In a second example, the protease ompT was used and led to an enrichment of the known double-arginine motif. The IMOP system thus substantially improves and simplifies previous systems.

MeSH terms

  • Peptide Hydrolases / chemistry*
  • Peptide Library*
  • Serine Endopeptidases / chemistry
  • Serine Endopeptidases / metabolism
  • Substrate Specificity
  • Subtilisin / chemistry
  • Subtilisin / metabolism

Substances

  • Peptide Library
  • Peptide Hydrolases
  • Serine Endopeptidases
  • Subtilisin
  • omptin outer membrane protease