Functional Ca2+ channel produced by purified platelet membrane glycoprotein IIB-IIIA complex incorporated into planar phospholipid bilayer

Thromb Haemost. 1991 Nov 1;66(5):598-603.

Abstract

The ability of the platelet membrane glycoprotein (GP) IIb-IIIa complex to function as a Ca2+ channel was investigated by electrophysiological methods. The GPIIb-IIIa complex was purified with an electrically silent detergent, CHAPS, and reconstituted into liposomes. After incorporation of these liposomes to a planar phospholipid bilayer, Ba(2+)-permeable channel currents were detected. Since neither residual detergent nor dissociated GPIIb and IIIa produced any currents, the observed channel currents were attributed to the GPIIb-IIIa complex. These channel currents showed similar electrical properties with the Ca2+ channel previously described in platelet plasma membrane; a single channel conductance of approximately 10 pS in 53 mM Ba2+ solution and voltage-independency. It was concluded that the purified GPIIb-IIIa complex can act as a divalent cation-permeable channel in the artificial phospholipid bilayer.

Publication types

  • Comparative Study
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Calcium Channels / physiology*
  • Electrophoresis, Polyacrylamide Gel
  • Electrophysiology / instrumentation
  • Electrophysiology / methods
  • Humans
  • Lipid Bilayers*
  • Membrane Potentials
  • Platelet Membrane Glycoproteins / isolation & purification
  • Platelet Membrane Glycoproteins / physiology*
  • Structure-Activity Relationship
  • Thrombin / pharmacology

Substances

  • Calcium Channels
  • Lipid Bilayers
  • Platelet Membrane Glycoproteins
  • Thrombin