Altered endothelin-1 vasoreactivity in patients with untreated normal-pressure glaucoma

Invest Ophthalmol Vis Sci. 2006 Jun;47(6):2528-32. doi: 10.1167/iovs.05-0240.

Abstract

Purpose: Vasospasm, resulting from a generalized dysfunction in the vascular endothelium, is implicated in the development of normal-pressure glaucoma (NPG). Impaired endothelium-derived nitric oxide activity and abnormalities of the endothelin system suggest systemic endothelial cell dysfunction in patients with NPG. Endothelin (ET)-1 vasoreactivity was assessed in the peripheral circulation of patients with NPG.

Methods: Forearm blood flow was measured using venous occlusion plethysmography in eight patients with untreated NPG and eight age- and sex-matched healthy volunteers during intra-arterial infusion of ET-1 (5 pmol/min) and, on a separate occasion, to BQ123, a selective endothelin-A receptor antagonist, (100 nmol/min). Blood pressure and heart rate were measured in the noninfused arm, and plasma ET-1 concentrations were measured using a radioimmunoassay.

Results: Forearm blood flow fell during infusion of ET-1 (P<0.001 for both) to a similar extent in both groups (P=0.7; patients versus control subjects). In contrast, BQ123 increased forearm blood flow in both groups (P<0.001 for both), although the vasodilatation was lower in patients than in control subjects (P<0.001; patients versus control subjects). There was no difference in basal plasma ET-1 concentrations between the two groups (P=0.81; patients versus control subjects).

Conclusions: Despite normal responses to ET-1, patients with NPG have reduced vasodilatation in response to ETA-receptor antagonism. This could be due to attenuated ETA-receptor-mediated tone, increased ETB-receptor-mediated contraction or impaired ETB-receptor-mediated release of endothelial nitric oxide. These results are consistent with the authors' previous demonstration of systemic vascular dysfunction in patients with NPG.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Blood Flow Velocity
  • Blood Pressure
  • Endothelin A Receptor Antagonists
  • Endothelin-1 / administration & dosage
  • Endothelin-1 / blood
  • Endothelin-1 / physiology*
  • Endothelium, Vascular / physiology
  • Female
  • Forearm / blood supply
  • Glaucoma, Open-Angle / blood
  • Glaucoma, Open-Angle / physiopathology*
  • Heart Rate
  • Humans
  • Intraocular Pressure*
  • Male
  • Middle Aged
  • Peptides, Cyclic / administration & dosage
  • Radioimmunoassay
  • Vasodilation / physiology*

Substances

  • Endothelin A Receptor Antagonists
  • Endothelin-1
  • Peptides, Cyclic
  • cyclo(Trp-Asp-Pro-Val-Leu)