Biochemical and biological characterization of a neuroendocrine-associated phosphatase

J Neurochem. 2006 Jul;98(1):89-101. doi: 10.1111/j.1471-4159.2006.03852.x.

Abstract

The biochemical and biological properties of a novel neuroendocrine-associated phosphatase (NEAP) were characterized. NEAP had a sequence characteristic of a dual-specificity phosphatase (DSP), and was preferentially expressed in neuroendocrine cells/tissues as well as in skeletal muscle and heart. Expression of NEAP was up-regulated in nerve growth factor (NGF)-treated, differentiated PC12 cells. NEAP was cytosolic and did not apparently have effects against extracellular signal-regulated kinase, c-Jun N-terminal kinase (JNK) and p38 mitogen-activated protein kinase activated by various stimuli. Although NEAP and MAPK phosphatase (MPK)-1 showed similar phosphatase activity towards p-nitro phenylphosphate (pNPP), in contrast to MKP-1, NEAP did not dephosphorylate JNK and p38-MAPK in vitro. Overexpression of NEAP, but not the C152S mutant, in PC12 cells suppressed NGF-induced phosphorylation of the p85 subunit of phosphatidylinositol 3-kinase (PI3K) and Akt activation. Overexpression of NEAP also suppressed neurite outgrowth induced by NGF and sensitized PC12 cells to cisplatin-induced apoptosis. Suppression of NEAP by RNA interference enhanced NGF-induced neurite outgrowth and Akt activation. Our results indicated that, unlike other DSPs, down-regulation of conventional MAPKs was not the major function of NEAP. Furthermore, NEAP might be involved in neuronal differentiation via regulation of the PI3K/Akt signaling.

Publication types

  • Comparative Study
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Cell Differentiation / drug effects
  • Cell Differentiation / physiology*
  • Cell Fractionation / methods
  • Cell Line
  • Dose-Response Relationship, Drug
  • Dual-Specificity Phosphatases
  • Enzyme Activation / drug effects
  • Enzyme Activation / physiology
  • Gene Expression / drug effects
  • Humans
  • Immunoprecipitation / methods
  • Mitogen-Activated Protein Kinase Phosphatases
  • Mitogen-Activated Protein Kinases / metabolism
  • Mutation / physiology
  • Nerve Growth Factor / pharmacology
  • Neurons / drug effects
  • Neurons / physiology
  • Neurosecretory Systems / cytology
  • Neurosecretory Systems / metabolism*
  • Phosphoric Monoester Hydrolases / chemistry
  • Phosphoric Monoester Hydrolases / physiology*
  • RNA, Messenger / metabolism
  • Rats
  • Reverse Transcriptase Polymerase Chain Reaction / methods
  • Sequence Alignment / methods
  • Signal Transduction / drug effects
  • Signal Transduction / physiology*
  • Time Factors
  • Transfection / methods

Substances

  • RNA, Messenger
  • Nerve Growth Factor
  • Mitogen-Activated Protein Kinases
  • Mitogen-Activated Protein Kinase Phosphatases
  • Phosphoric Monoester Hydrolases
  • DUSP26 protein, human
  • Dual-Specificity Phosphatases