Differential effects of oral conjugated equine estrogen and transdermal estrogen on atherosclerotic vascular disease risk markers and endothelial function in healthy postmenopausal women

Hum Reprod. 2006 Oct;21(10):2715-20. doi: 10.1093/humrep/del245. Epub 2006 Jun 28.

Abstract

Background: Recent studies have revealed that HRT may increase the risk for atherosclerotic vascular disease (ASVD).

Methods: We investigated the effects of HRT via different administration routes on the markers for ASVD and endothelial function in healthy postmenopausal women. The oral HRT group (n=18) received conjugated equine estrogen 0.625 mg/day; the transdermal HRT group (n=18) received 17beta-estradiol (E2) gel 0.6 mg/day for 6 months. The control group (n=30) had no treatment for 6 months.

Results: The C-reactive protein (CRP) rose from 0.129+/-0.116 to 0.752+/-0.794 mg/dl (P<0.01) in the oral HRT group but remained unchanged in the transdermal HRT and control groups. The flow-mediated vasodilation (FMD) in the brachial artery was increased significantly by HRT from 6.0% before oral HRT to 14.7% after oral HRT (P<0.001) and from 5.9% before transdermal HRT to 13.9% after transdermal HRT (P=0.001).

Conclusions: These data suggest that oral estrogen induces ASVD risk by increasing acute inflammation; however, transdermal estrogen avoids this untoward effect. Additionally, transdermal estrogen exerts a positive effect on endothelial function similar to that of oral estrogen. Therefore, the transdermal route might be favourable in terms of ASVD risks.

Publication types

  • Controlled Clinical Trial
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Administration, Oral
  • Aged
  • Atherosclerosis / prevention & control*
  • Biomarkers
  • Brachial Artery / drug effects
  • Brachial Artery / physiology*
  • Estrogen Replacement Therapy
  • Estrogens / administration & dosage
  • Estrogens / therapeutic use*
  • Estrogens, Conjugated (USP) / administration & dosage
  • Estrogens, Conjugated (USP) / therapeutic use*
  • Female
  • Follicle Stimulating Hormone / blood
  • Hormones / blood
  • Humans
  • Hysterectomy
  • Lipids / blood
  • Middle Aged
  • Postmenopause / drug effects
  • Postmenopause / physiology*
  • Vasodilation / drug effects*

Substances

  • Biomarkers
  • Estrogens
  • Estrogens, Conjugated (USP)
  • Hormones
  • Lipids
  • Follicle Stimulating Hormone