Release of cholecystokinin from rat midbrain slices and modulatory effect of D2DA receptor stimulation

Brain Res. 1991 Aug 2;555(2):281-7. doi: 10.1016/0006-8993(91)90353-w.

Abstract

Cholecystokinin octapeptide (CCK-8) is colocalized within a majority of dopamine (DA)-containing neurons of the rat midbrain. Exogenous CCK-8 can modulate the electrophysiological activity of DA neurons, at least in part, by direct actions on the somatodendritic region of these cells. If CCK-8 is somatodendritically released from DA neurons, it may influence DA cell function as has been shown for DA itself. In the present study, radioimmunoassay was used to determine if CCK-8 is released in vitro from slices of rat midbrain under basal and depolarizing (30 mM potassium) conditions. Low levels of CCK-8 were detected in the basal incubation medium. Thirty mM potassium caused about a 3-fold increase in the release of CCK-8. This stimulated release was abolished in calcium-free medium. The D2 receptor agonist quinpirole, but not the D1 agonist SKF 38393, attenuated the potassium-stimulated release of CCK-8 but did not affect basal release. These results show that CCK-8, like DA, can be released from midbrain slices, presumably from DA/CCK-8-containing neurons. This finding is in accordance with the possibility that CCK-8 plays a role in the regulation of DA neuronal function at the level of the cell body, where it might influence the excitability of the DA cell membrane.

Publication types

  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine / pharmacology
  • Animals
  • Cholecystokinin / immunology
  • Cholecystokinin / metabolism*
  • Chromatography, High Pressure Liquid
  • Dopamine Agents / pharmacology
  • Ergolines / pharmacology
  • In Vitro Techniques
  • Iodine Radioisotopes
  • Male
  • Mesencephalon / metabolism*
  • Potassium / pharmacology
  • Quinpirole
  • Radioimmunoassay
  • Rats
  • Rats, Inbred Strains
  • Receptors, Dopamine / drug effects
  • Receptors, Dopamine / metabolism*
  • Receptors, Dopamine D1
  • Receptors, Dopamine D2
  • Sulpiride / pharmacology
  • Veratridine / pharmacology

Substances

  • Dopamine Agents
  • Ergolines
  • Iodine Radioisotopes
  • Receptors, Dopamine
  • Receptors, Dopamine D1
  • Receptors, Dopamine D2
  • Quinpirole
  • 2,3,4,5-Tetrahydro-7,8-dihydroxy-1-phenyl-1H-3-benzazepine
  • Veratridine
  • Sulpiride
  • Cholecystokinin
  • Potassium