Bradykinin is a potent pruritogen in atopic dermatitis: a switch from pain to itch

Pain. 2006 Dec 15;126(1-3):16-23. doi: 10.1016/j.pain.2006.06.003. Epub 2006 Jul 13.

Abstract

Histamine, substance P, serotonin and bradykinin were applied by iontophoresis to lesional and visually non-lesional skin of 14 patients with atopic dermatitis, and normal skin of 15 healthy volunteers. Itch could be evoked by light stroking of skin with a cotton swab (alloknesis) in all lesional skin sites, but not in non-lesional or normal skin. Substances were applied in the same skin area before and 3 h after administration of placebo or antihistamine (olopatadine hydrochloride: H1-receptor-blocker). Intensities of itch and pain sensation and areas of flare and wheal were measured. All the substances induced significantly more intense itch in lesional skin than in non-lesional skin of patients. Even bradykinin, which evoked only weak itch and pain of similar intensities in non-lesional skin of patients and in healthy volunteers, induced intense itch in lesional skin, while the simultaneously increased pain did not suppress the itch sensation, indicating central sensitization. Histamine- and substance P-induced itch was almost completely suppressed by antihistamines, whereas bradykinin- and serotonin-induced itch was not. This suggests that substance P is a histamine-dependent pruritogen also in lesional skin under sensitized conditions but that bradykinin and serotonin are histamine-independent pruritogens in lesional skin. It is concluded that serotonin and bradykinin, classic endogenous algogens, can turn into potent histamine-independent pruritogens in lesional skin of atopic dermatitis.

MeSH terms

  • Adult
  • Bradykinin / administration & dosage*
  • Cross-Over Studies
  • Dermatitis, Atopic / complications*
  • Female
  • Histamine / administration & dosage
  • Histamine H1 Antagonists / pharmacology
  • Humans
  • Iontophoresis
  • Male
  • Pain / etiology
  • Pruritus / chemically induced
  • Pruritus / etiology*
  • Pruritus / physiopathology
  • Serotonin / administration & dosage
  • Single-Blind Method
  • Substance P / administration & dosage
  • Urticaria / chemically induced
  • Water / administration & dosage

Substances

  • Histamine H1 Antagonists
  • Water
  • Serotonin
  • Substance P
  • Histamine
  • Bradykinin