In vitro inhibitory effect of antituberculosis drugs on clinical and environmental strains of Coccidioides posadasii

J Antimicrob Chemother. 2006 Sep;58(3):575-9. doi: 10.1093/jac/dkl290. Epub 2006 Jul 24.

Abstract

Objectives: The aim of the present study was to evaluate the in vitro effect of the first-line antimicrobial drugs for pulmonary tuberculosis against the fungal pathogen Coccidioides posadasii.

Methods: The in vitro activities of rifampicin, isoniazid, pyrazinamide and ethambutol against clinical and environmental strains of C. posadasii were determined in accordance with the CSLI M38-A macrodilution method. The antimicrobials were tested alone or in combinations of two or more drugs.

Results: With the exception of pyrazinamide, all of the tested drugs interfered with the in vitro growth of C. posadasii. The 2 day MIC ranges of the tested drugs were as follows: rifampicin 1,060-4,250 mg/L; isoniazid < or =250 mg/L; ethambutol < or =620 mg/L. Pronounced in vitro synergism was demonstrated for combined antituberculosis drugs. The combination of rifampicin plus pyrazinamide was the only one that did not inhibit fungal growth.

Conclusions: The present study showed that the first-line antituberculosis drugs, alone or in combinations, interfered with the vegetative growth of C. posadasii strains in vitro. Further studies in a murine model will need to be conducted in order to evaluate the in vivo effect of antituberculosis drugs on Coccidioides spp.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Antifungal Agents / pharmacology*
  • Antitubercular Agents / pharmacology*
  • Coccidioides / drug effects*
  • Coccidioides / isolation & purification
  • Coccidioidomycosis / microbiology*
  • Drug Synergism
  • Humans
  • Microbial Sensitivity Tests
  • Time Factors

Substances

  • Antifungal Agents
  • Antitubercular Agents