Platelet 5-HT2A receptor subresponsivity and lethality of attempted suicide in depressed in-patients

Int J Neuropsychopharmacol. 2007 Jun;10(3):335-43. doi: 10.1017/S1461145706006997. Epub 2006 Aug 8.

Abstract

In depressed patients, high-lethality suicidal acts are accompanied by serotonin system abnormalities analogous to those seen in completed suicides. We have previously reported greater platelet 5-HT2A receptor density, and impaired serotonin enhancement of ADP-induced platelet aggregation, an indirect measure of signal transduction, in high-lethality suicide attempters. We hypothesized that serotonin-activated phosphoinositide (PI) hydrolysis, a direct measure of platelet serotonin 5-HT2A receptor responsivity would be lower in depressed high-lethality suicide attempters. Twenty-three depressed in-patients that had previously made suicide attempts (low-lethality, n=6; high-lethality, n=17) had platelet 5-HT2A-mediated serotonin-simulated PI hydrolysis assayed. Platelet 5-HT2A receptor responsivity in high-lethality suicide attempters was 41% that of low-lethality suicide attempters (p<0.05). A seasonal effect was also observed. High-lethality suicidal acts are associated with more 5-HT2A receptors but impaired signal transduction.

Publication types

  • Research Support, N.I.H., Extramural

MeSH terms

  • Adolescent
  • Adrenergic alpha-Agonists / pharmacology
  • Adult
  • Aged
  • Aged, 80 and over
  • Aging / psychology
  • Blood Platelets / metabolism*
  • Data Interpretation, Statistical
  • Depressive Disorder, Major / blood*
  • Depressive Disorder, Major / psychology*
  • Epinephrine / pharmacology
  • Female
  • Humans
  • Inpatients
  • Longitudinal Studies
  • Male
  • Middle Aged
  • Phosphatidylinositols / metabolism
  • Prefrontal Cortex / drug effects
  • Prefrontal Cortex / metabolism
  • Psychiatric Status Rating Scales
  • RNA, Messenger / biosynthesis
  • RNA, Messenger / genetics
  • Receptor, Serotonin, 5-HT2A / blood*
  • Receptors, Adrenergic, alpha-2 / drug effects
  • Seasons
  • Second Messenger Systems / genetics
  • Second Messenger Systems / physiology
  • Signal Transduction / physiology
  • Suicide / statistics & numerical data*
  • Suicide, Attempted / psychology*

Substances

  • Adrenergic alpha-Agonists
  • Phosphatidylinositols
  • RNA, Messenger
  • Receptor, Serotonin, 5-HT2A
  • Receptors, Adrenergic, alpha-2
  • Epinephrine