Classification of alpha-cyclodextrins inclusion complexes into Type 1 and Type 2: a prelude to log K prediction

J Mol Graph Model. 2007 Jan;25(5):731-9. doi: 10.1016/j.jmgm.2006.06.003. Epub 2006 Jun 17.

Abstract

Molecular Interaction Fields (MIFs) were used in combination with a small number of geometrical descriptors to separate nine alpha-CD complexes into Type 1 and Type 2, two classes, respectively, containing complexes having high log K and low log K values (stoichiometry of 1:1). Calculations were performed on the crystallographic conformations of alpha-CDs after their separation from the ligand and without minimization. The results show that the computational strategy adopted is able to distinguish Type 1 from Type 2 complexes and that it can be applied to all CD families.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Carbohydrate Conformation
  • Computer Graphics
  • Computer Simulation
  • Crystallography, X-Ray
  • Hydrophobic and Hydrophilic Interactions
  • Ligands
  • Macromolecular Substances
  • Models, Molecular
  • Thermodynamics
  • alpha-Cyclodextrins / chemistry*
  • alpha-Cyclodextrins / classification

Substances

  • Ligands
  • Macromolecular Substances
  • alpha-Cyclodextrins