Prostacyclin therapy increases right ventricular capillarisation in a model for flow-associated pulmonary hypertension

Eur J Pharmacol. 2006 Nov 7;549(1-3):107-16. doi: 10.1016/j.ejphar.2006.08.016. Epub 2006 Aug 17.

Abstract

Pulmonary hypertension, and consequently right ventricular failure, complicates several congenital heart defects. Although intervention in the prostacyclin-thromboxane ratio is known to improve outcome, the underlying mechanism is not clear. Therefore, effects of acetyl salicylic acid and iloprost are studied in an animal model for flow-associated pulmonary hypertension. Male Wistar rats with flow-associated pulmonary hypertension, an aortocaval shunt in addition to monocrotaline induced pulmonary hypertension, were treated with low-dose aspirin (25 mg/kg/day) or iloprost (72 microg/kg/day). Effects on pulmonary hemodynamics and pulmonary vascular remodeling as well as right ventricular hemodynamics and remodeling were evaluated. Ninety percent (n=7/8) of the untreated pulmonary hypertensive rats developed dyspnea and pleural fluid, whereas this was seen in 50% (n=4/8, ns) and 10% (n=1/8, P<0.05 vs. untreated animals) of the aspirin and iloprost-treated rats, respectively. This could not be attributed to changes in pulmonary artery pressure, wall-lumen ratio of the pulmonary vasculature or right ventricular hypertrophy. However, both therapies restored reduced right ventricular capillary to myocyte ratio in pulmonary hypertensive rats (0.95+/-0.10 in untreated rats vs. 1.38+/-0.18 in control animals; P<0.05, and 1.32+/-0.11 in aspirin-treated and 1.29+/-0.9 in iloprost-treated rats; both P<0.05 vs. non-treated animals), which was associated with improved right ventricular contractility (iloprost). Thus, interventions in the prostacyclin-thromboxane metabolism improve outcome in rats with flow-associated pulmonary hypertension. However, these effects may be attributed to effects on cardiac rather than on pulmonary vascular remodeling.

MeSH terms

  • Animals
  • Arachidonic Acid / metabolism
  • Aspirin / therapeutic use*
  • Blood Pressure / drug effects
  • Capillaries / drug effects
  • Capillaries / physiopathology
  • Disease Models, Animal
  • Echocardiography
  • Gene Expression / drug effects
  • Heart Ventricles / drug effects*
  • Heart Ventricles / metabolism
  • Heart Ventricles / physiopathology
  • Hypertension, Pulmonary / drug therapy*
  • Hypertension, Pulmonary / mortality
  • Hypertension, Pulmonary / physiopathology
  • Iloprost / therapeutic use*
  • Lung / blood supply
  • Lung / pathology
  • Lung / physiopathology
  • Male
  • Myocardium / pathology
  • Organ Size / drug effects
  • Platelet Aggregation Inhibitors / therapeutic use
  • Pulmonary Artery / drug effects
  • Pulmonary Artery / physiopathology
  • Pulmonary Circulation / drug effects
  • Rats
  • Rats, Wistar
  • Receptors, Vascular Endothelial Growth Factor / genetics
  • Survival Rate
  • Vascular Endothelial Growth Factor A / genetics
  • Ventricular Remodeling / drug effects

Substances

  • Platelet Aggregation Inhibitors
  • Vascular Endothelial Growth Factor A
  • Arachidonic Acid
  • Receptors, Vascular Endothelial Growth Factor
  • Iloprost
  • Aspirin