Improvement in rod and cone function in mouse model of Fundus albipunctatus after pharmacologic treatment with 9-cis-retinal

Invest Ophthalmol Vis Sci. 2006 Oct;47(10):4540-6. doi: 10.1167/iovs.06-0215.

Abstract

Purpose: To assess changes in rod and cone visual functions in a mouse model of Fundus albipunctatus with disrupted 11-cis-retinol dehydrogenase (RDH) genes after pharmacologic treatment with an artificial retinal chromophore.

Methods: Retinoid levels and photoreceptor functions of Rdh5-/-Rdh11-/- mice at a variety of light intensities were analyzed with normal-phase HPLC and ERG techniques. Production of 11-cis-retinal, the visual pigment chromophore, was suppressed with a potent inhibitor of the retinoid cycle, all-trans-retinylamine (Ret-NH2). The chromophore was replaced by a functional geometric isomer, 9-cis-retinal, delivered by oral gavage.

Results: Aberrant cone responses were detected in 12-month-old Rdh5-/-Rdh11-/- mice raised in a 12-hour light/12-hour dark cycle. This cone defect was exacerbated in conditions of low levels of 11-cis-retinal. Administration of 9-cis-retinal increased the rate of dark adaptation and improved cone function in Rdh5-/-Rdh11-/- mice.

Conclusions: Disruption of 11-cis-RDHs causes a slowly developing cone dystrophy caused by inefficient cone pigment regeneration. Rod and cone visual function improved significantly in the mouse model of F. albipunctatus after treatment with 9-cis-retinal, suggesting a potential approach to slow the progression of cone dystrophy in affected humans.

Publication types

  • Research Support, N.I.H., Extramural

MeSH terms

  • Animals
  • Chromatography, High Pressure Liquid
  • Dark Adaptation
  • Disease Models, Animal*
  • Diterpenes
  • Electroretinography
  • Isomerism
  • Mice
  • Mice, Knockout
  • Oxidoreductases / physiology
  • Photoreceptor Cells, Vertebrate / physiology*
  • Pigment Epithelium of Eye / physiology
  • Retinal Degeneration / drug therapy*
  • Retinal Degeneration / metabolism
  • Retinal Degeneration / physiopathology
  • Retinal Dehydrogenase / physiology
  • Retinaldehyde / therapeutic use*
  • Retinoids / metabolism

Substances

  • Diterpenes
  • Retinoids
  • 9-cis-retinal
  • Oxidoreductases
  • Rdh11 protein, mouse
  • Retinal Dehydrogenase
  • Retinaldehyde