Rotigotine for the treatment of Parkinson's disease

Expert Rev Neurother. 2006 Sep;6(9):1275-82. doi: 10.1586/14737175.6.9.1275.

Abstract

Dopaminergic therapies, including levodopa and dopamine agonists, are the mainstays of therapy in Parkinson's disease. With the exception of the injectable short-acting dopamine agonist apomorphine, there is no other widely available non-oral dopaminergic therapy. Rotigotine is a lipid-soluble, non-ergot, D3, D2, D1 dopamine receptor agonist that has demonstrated efficacy as an alternative therapeutic option in both early and advanced Parkinson's disease. More importantly, it is uniquely formulated as a transdermal patch delivery system allowing for continuous, once-daily administration and better patient compliance. Preclinical and clinical trials have shown rotigotine to be a well-tolerated and effective treatment for early-stage Parkinson's disease. Rotigotine has also shown promise as adjunctive therapy with levodopa for the treatment of advanced Parkinson's disease.

Publication types

  • Review

MeSH terms

  • Antiparkinson Agents / administration & dosage
  • Antiparkinson Agents / adverse effects
  • Clinical Trials as Topic*
  • Humans
  • Parkinson Disease / drug therapy*
  • Practice Patterns, Physicians' / trends
  • Tetrahydronaphthalenes / administration & dosage*
  • Tetrahydronaphthalenes / adverse effects
  • Thiophenes / administration & dosage*
  • Thiophenes / adverse effects

Substances

  • Antiparkinson Agents
  • Tetrahydronaphthalenes
  • Thiophenes
  • rotigotine