Alkali pH directly activates ATP-sensitive K+ channels and inhibits insulin secretion in beta-cells

Biochem Biophys Res Commun. 2006 Nov 17;350(2):492-7. doi: 10.1016/j.bbrc.2006.09.084. Epub 2006 Sep 26.

Abstract

Glucose stimulation of pancreatic beta-cells is reported to lead to sustained alkalization, while extracellular application of weak bases is reported to inhibit electrical activity and decrease insulin secretion. We hypothesize that beta-cell K(ATP) channel activity is modulated by alkaline pH. Using the excised patch-clamp technique, we demonstrate a direct stimulatory action of alkali pH on recombinant SUR1/Kir6.2 channels due to increased open probability. Bath application of alkali pH similarly activates native islet beta-cell K(ATP) channels, leading to an inhibition of action potentials, and hyperpolarization of membrane potential. In situ pancreatic perfusion confirms that these cellular effects of alkali pH are observable at a functional level, resulting in decreases in both phase 1 and phase 2 glucose-stimulated insulin secretion. Our data are the first to report a stimulatory effect of a range of alkali pH on K(ATP) channel activity and link this to downstream effects on islet beta-cell function.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • ATP-Binding Cassette Transporters / metabolism*
  • Adenosine Triphosphate / metabolism
  • Alkalies / chemistry
  • Animals
  • Hydrogen-Ion Concentration
  • Insulin / metabolism*
  • Insulin Secretion
  • Insulin-Secreting Cells / metabolism
  • Insulin-Secreting Cells / physiology*
  • Male
  • Membrane Potentials
  • Mice
  • Patch-Clamp Techniques
  • Potassium Channels / metabolism*
  • Potassium Channels, Inwardly Rectifying / metabolism*
  • Rats
  • Rats, Wistar
  • Receptors, Drug / metabolism*
  • Sulfonylurea Receptors

Substances

  • ATP-Binding Cassette Transporters
  • Abcc8 protein, mouse
  • Abcc8 protein, rat
  • Alkalies
  • Insulin
  • Kir6.2 channel
  • Potassium Channels
  • Potassium Channels, Inwardly Rectifying
  • Receptors, Drug
  • Sulfonylurea Receptors
  • Adenosine Triphosphate