Characterization of the androgen receptor in a benign prostate tissue-derived human prostate epithelial cell line: RC-165N/human telomerase reverse transcriptase

Prostate Cancer Prostatic Dis. 2007;10(1):30-8. doi: 10.1038/sj.pcan.4500915. Epub 2006 Oct 31.

Abstract

The majority of prostate epithelial cell lines stably expressing wild-type (wt) or mutant (mt) androgen receptor (AR) are derived from metastatic prostate cancers. Therefore, the wt AR-expressing RC-165N/human telomerase reverse transcriptase (hTERT) cell line derived from the benign prostate tissue of an African-American patient provides a unique opportunity to assess the functional status of AR in a cellular context not studied before. Although androgen-induced expression of known androgen responsive genes such as PMEPA1, and NDRG1 was observed in RC-165N/hTERT, this cell line expresses prostate-specific antigen (PSA) at significantly lower levels. Chromatin immunoprecipitation assay revealed androgen-dependent binding of AR to androgen response elements of PSA, PMEPA1 and NDRG1 genes. Similarities, as well as differences were noted in the expression of androgen responsive genes between RC-165N/hTERT and LNCaP cells. Comprehensive evaluations of AR functions in RC-165N/hTERT cells suggest that whereas some features of known AR functions are maintained in this benign prostatic tissue-derived cell line, other AR functions are not retained. Objective evaluations of similar cell lines will lead to the understanding of AR functions in prostate growth and differentiation.

Publication types

  • Research Support, Non-U.S. Gov't
  • Research Support, U.S. Gov't, Non-P.H.S.

MeSH terms

  • Cell Line, Transformed
  • Cluster Analysis
  • Dihydrotestosterone / pharmacology
  • Epithelial Cells / metabolism*
  • Gene Expression Regulation / drug effects
  • Humans
  • Male
  • Oligonucleotide Array Sequence Analysis
  • Prostate-Specific Antigen / metabolism
  • Prostatic Hyperplasia / genetics
  • Prostatic Hyperplasia / metabolism*
  • Prostatic Hyperplasia / pathology
  • Receptors, Androgen / metabolism*
  • Receptors, Androgen / physiology
  • Response Elements
  • Telomerase / genetics*

Substances

  • Receptors, Androgen
  • Dihydrotestosterone
  • Telomerase
  • Prostate-Specific Antigen