Gefitinib efficacy associated with multiple expression of HER family in non-small cell lung cancer

Anticancer Res. 2006 Sep-Oct;26(5B):3761-5.

Abstract

The aim of this study was to compare the relationship between HER family expression and clinical response to gefitinib.

Patients and methods: Tissues from thirty-one non-small cell lung cancer (NSCLC) patients treated with a monotherapy of gefitinib were analyzed. Expressions of HER family in 31 tumors were examined by immunohistochemistry.

Results: The total expressions were 21 for EGFR (68%), 24 for HER2 (77%), 17 for HER3 (55%) and 4 for HER4 (13%). Fourteen out of 31 (45%) demonstrated triple expression of EGFR and HER2, as well as HER3 or HER4. A significantly better response rate (RR) and time to progression (TTP) were observed for the group with the triple expression than for the other groups (RR 50 vs. 11%; p < 0.05, median TTP 4.29 vs. 1.2 months; p < 0.05).

Conclusion: Mutliple expression of the HER family might be related with the clinical response to gefitinib and EGFR mutation status.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Aged
  • Antineoplastic Agents / therapeutic use*
  • Base Sequence
  • Carcinoma, Non-Small-Cell Lung / drug therapy*
  • Carcinoma, Non-Small-Cell Lung / metabolism
  • DNA Primers
  • Disease Progression
  • ErbB Receptors / genetics
  • Female
  • Gefitinib
  • Humans
  • Lung Neoplasms / drug therapy*
  • Lung Neoplasms / metabolism
  • Male
  • Middle Aged
  • Mutation
  • Quinazolines / therapeutic use*
  • Receptor Protein-Tyrosine Kinases / metabolism*
  • Survival Analysis

Substances

  • Antineoplastic Agents
  • DNA Primers
  • Quinazolines
  • ErbB Receptors
  • Receptor Protein-Tyrosine Kinases
  • Gefitinib