Mucin 1 oncoprotein blocks hypoxia-inducible factor 1alpha activation in a survival response to hypoxia

J Biol Chem. 2007 Jan 5;282(1):257-66. doi: 10.1074/jbc.M610156200. Epub 2006 Nov 13.

Abstract

Resistance of carcinoma cells to hypoxic stress is of importance to the growth of solid tumors. The mucin 1 (MUC1) oncoprotein is aberrantly overexpressed by most human carcinomas; however, there is no known relationship between MUC1 and the hypoxic stress response. The present work has demonstrated that MUC1 attenuates activation of hypoxia-inducible factor-1alpha (HIF-1alpha), a regulator of gene transcription in the response of cells to hypoxic stress. In cells with stable gain and loss of MUC1 function, we have shown that MUC1 up-regulates prolyl hydroxylase 3 (PHD3) expression and promotes HIF-1alpha degradation. PHD activity is attenuated by increases in reactive oxygen species (ROS) generated in the hypoxic stress response. Our results further demonstrate that MUC1 blocks hypoxia-induced increases in ROS and thereby potentiates PHD-mediated HIF-1alpha suppression. Importantly, MUC1 also blocks hypoxia-induced apoptosis and necrosis by suppressing accumulation of ROS. These findings indicate that MUC1 attenuates HIF-1alpha activation in a survival response to hypoxic stress.

Publication types

  • Research Support, N.I.H., Extramural

MeSH terms

  • Apoptosis
  • Cell Line, Tumor
  • Gene Expression Regulation, Neoplastic*
  • Gene Silencing
  • Humans
  • Hypoxia*
  • Hypoxia-Inducible Factor 1, alpha Subunit / chemistry*
  • Hypoxia-Inducible Factor 1, alpha Subunit / metabolism
  • Mitochondria / metabolism
  • Mucin-1 / chemistry*
  • Necrosis
  • Oncogene Proteins / chemistry*
  • Procollagen-Proline Dioxygenase / metabolism
  • Protein Structure, Tertiary
  • Reactive Oxygen Species
  • Up-Regulation

Substances

  • HIF1A protein, human
  • Hypoxia-Inducible Factor 1, alpha Subunit
  • Mucin-1
  • Oncogene Proteins
  • Reactive Oxygen Species
  • Procollagen-Proline Dioxygenase