Edaravone protects the vestibular periphery from free radical-induced toxicity in response to perilymphatic application of (+/-)-alpha-amino-3-hydroxy-5-methyl-isoxazole-4-propionic acid

Eur J Pharmacol. 2007 Jan 12;554(2-3):223-8. doi: 10.1016/j.ejphar.2006.10.030. Epub 2006 Oct 20.

Abstract

Intracochlear infusion of (+/-)-alpha-amino-3-hydroxy-5-methyl-isoxazole-4-propionic acid (AMPA) was performed with a syringe pump in guinea pigs, and peripheral vestibular dysfunction was induced. Animals were administered edaravone systemically or topically. In the systemic application group, animals were administered edaravone once a day for 7 days after AMPA infusion. In the topical application group, edaravone-soaked gelfoam was placed on the round window membrane just after, 12 h after or 24 h after AMPA infusion. Spontaneous nystagmus was observed after AMPA infusion. Immunohistochemistry for 4-hydroxy-2-nonenal (4-HNE), a marker of free radical-induced lipid peroxidation, was performed 24 h after AMPA infusion. In addition, caloric tests were performed to evaluate vestibular function 1 week after AMPA infusion. Animals in both groups showed decreased spontaneous nystagmus, but results were not significant. Animals treated topically with edaravone within 12 h of AMPA infusion showed normal morphology of the ampullar sensory epithelia of the lateral semicircular canals and showed a good response to the caloric tests. 4-HNE immunoreactivity in the sensory epithelia was very low in these animals. In contrast, untreated animals and animals treated with edaravone systemically or topically 24 h after AMPA infusion showed morphologic hair cell damage, reduced caloric response and remarkable 4-HNE immunoreactivity in the sensory epithelia. These results indicate that topical application of edaravone within 12 h after damage protects the vestibular periphery from free radical-induced toxicity in response to intracochlear infusion of AMPA.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Aldehydes / metabolism
  • Animals
  • Antipyrine / analogs & derivatives*
  • Antipyrine / pharmacology
  • Edaravone
  • Excitatory Amino Acid Agonists / administration & dosage
  • Excitatory Amino Acid Agonists / toxicity
  • Free Radical Scavengers / pharmacology
  • Free Radicals / antagonists & inhibitors
  • Free Radicals / metabolism*
  • Guinea Pigs
  • Immunohistochemistry
  • Infusion Pumps
  • Male
  • Nystagmus, Pathologic / chemically induced
  • Nystagmus, Pathologic / physiopathology
  • Nystagmus, Pathologic / prevention & control
  • Reflex, Vestibulo-Ocular / drug effects
  • Vestibular Diseases / chemically induced
  • Vestibular Diseases / physiopathology
  • Vestibular Diseases / prevention & control*
  • Vestibular Function Tests
  • Vestibule, Labyrinth / drug effects*
  • Vestibule, Labyrinth / metabolism
  • Vestibule, Labyrinth / pathology
  • alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid / administration & dosage
  • alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid / toxicity*

Substances

  • Aldehydes
  • Excitatory Amino Acid Agonists
  • Free Radical Scavengers
  • Free Radicals
  • alpha-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid
  • 4-hydroxy-2-nonenal
  • Edaravone
  • Antipyrine