"Similarity trap" in protein-protein interactions could be carcinogenic: simulations of p53 core domain complexed with 53BP1 and BRCA1 BRCT domains

Structure. 2006 Dec;14(12):1811-21. doi: 10.1016/j.str.2006.10.009.

Abstract

Similar binding sites often imply similar protein-protein interactions and similar functions; however, similar binding sites may also constitute traps for nonfunctional associations. How are similar sites distinguished to prevent misassociations? BRCT domains from breast cancer-susceptibility gene product BRCA1 and protein 53BP1 have similar structures yet different binding behaviors with p53 core domain. 53BP1-BRCT domain forms a stable complex with p53. In contrast, BRCA1-p53 interaction is weak or other mechanisms operate. To delineate the difference, we designed 13 BRCA1-BRCT mutants and computationally investigated the structural and stability changes compared to the experimental p53-53BP1 structure. Interestingly, of the 13, the 2 mutations that are cancerous and involve nonconserved residues are those that enforced p53 core domain binding with BRCA1-BRCT in a way similar to p53-53BP1 binding. Hence, falling into the "similarity trap" may disrupt normal BRCA1 and p53 functions. Our results illustrate how this trap is avoided in the native state.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, N.I.H., Intramural

MeSH terms

  • Amino Acid Sequence
  • BRCA1 Protein / chemistry*
  • Binding Sites
  • Computer Simulation
  • Humans
  • Intracellular Signaling Peptides and Proteins / chemistry*
  • Models, Molecular
  • Molecular Sequence Data
  • Mutation
  • Phosphoproteins / chemistry*
  • Protein Binding
  • Protein Interaction Mapping / methods*
  • Protein Structure, Secondary
  • Protein Structure, Tertiary
  • Thermodynamics
  • Tumor Suppressor Protein p53 / chemistry*
  • Tumor Suppressor p53-Binding Protein 1

Substances

  • BRCA1 Protein
  • Intracellular Signaling Peptides and Proteins
  • Phosphoproteins
  • TP53 protein, human
  • TP53BP1 protein, human
  • Tumor Suppressor Protein p53
  • Tumor Suppressor p53-Binding Protein 1