Travoprost 0.004% with and without benzalkonium chloride: a comparison of safety and efficacy

J Glaucoma. 2007 Jan;16(1):98-103. doi: 10.1097/01.ijg.0000212274.50229.c6.

Abstract

Purpose: To compare the safety and efficacy of travoprost 0.004% without benzalkonium chloride (BAC) to that of the marketed formulation of travoprost 0.004% in patients with open-angle glaucoma or ocular hypertension.

Methods: The study was a double-masked, randomized, parallel group, multicenter, noninferiority design. Adult patients with open-angle glaucoma or ocular hypertension with qualifying intraocular pressure (IOP) on 2 eligibility visits received either travoprost 0.004% with BAC (n=346), or travoprost 0.004% without BAC (n=344) dosed once-daily each evening. Patients were followed for a period of 3 months. IOP measurements at 8 AM, 10 AM, and 4 PM were taken at study visits on week 2, week 6, and month 3.

Results: Mean IOP reductions, across all 9 study visits and times ranged from 7.3 to 8.5 mm Hg for travoprost 0.004% without BAC and from 7.4 to 8.4 mm Hg for travoprost 0.004% with BAC. Statistical equivalence was also demonstrated for the comparison of mean IOP changes; 95% confidence limits were within +/-0.8 mm Hg at 9 of 9 study visits and times in both the per protocol and intent-to-treat data sets. Adverse events and the number of patients discontinued owing to adverse events were similar for both treatment groups. Adverse events due to hyperemia occurred in 6.4% and 9.0% of patients treated with travoprost 0.004% without BAC and travoprost 0.004% with BAC, respectively.

Conclusion: Travoprost 0.004% without BAC is equivalent to travoprost 0.004% with BAC in both safety and efficacy.

Publication types

  • Comparative Study
  • Multicenter Study
  • Randomized Controlled Trial
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Aged
  • Antihypertensive Agents / administration & dosage*
  • Antihypertensive Agents / adverse effects
  • Antihypertensive Agents / therapeutic use
  • Benzalkonium Compounds / administration & dosage*
  • Benzalkonium Compounds / adverse effects
  • Benzalkonium Compounds / therapeutic use
  • Chemistry, Pharmaceutical
  • Cloprostenol / administration & dosage
  • Cloprostenol / adverse effects
  • Cloprostenol / analogs & derivatives*
  • Cloprostenol / therapeutic use
  • Double-Blind Method
  • Female
  • Glaucoma, Open-Angle / drug therapy*
  • Gonioscopy
  • Humans
  • Intraocular Pressure / drug effects*
  • Male
  • Middle Aged
  • Ocular Hypertension / drug therapy
  • Ophthalmic Solutions / administration & dosage
  • Ophthalmic Solutions / adverse effects
  • Ophthalmic Solutions / therapeutic use
  • Preservatives, Pharmaceutical / administration & dosage*
  • Preservatives, Pharmaceutical / adverse effects
  • Preservatives, Pharmaceutical / therapeutic use
  • Tonometry, Ocular
  • Travoprost
  • Treatment Outcome

Substances

  • Antihypertensive Agents
  • Benzalkonium Compounds
  • Ophthalmic Solutions
  • Preservatives, Pharmaceutical
  • Cloprostenol
  • Travoprost