A biosynthetically-inspired synthesis of the tetrahydrofuran core of obtusallenes II and IV

Org Lett. 2007 Feb 1;9(3):445-8. doi: 10.1021/ol062818g.

Abstract

[reaction: see text] Sharpless asymmetric dihydroxylation was regioselective for the trans olefin in an E vs Z vs terminal triene substrate. To test a biosynthetic hypothesis, the resulting diol underwent diastereoselective bromoetherification to provide the des-chloro core of marine natural products obtusallenes II and IV. Alternatively, anionic chloride ring-opening of a Z-beta,gamma-unsaturated epoxide gave separable regioisomeric halohydrins. Bromoetherification gave the fully elaborated core of obtusallenes II and IV with all of the relative stereochemistry correctly set.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Biological Products / chemistry*
  • Bromine / chemistry
  • Epoxy Compounds / chemistry
  • Ethers / chemistry
  • Furans / chemical synthesis*
  • Hydroxylation
  • Laurencia / chemistry*
  • Marine Biology*
  • Models, Chemical
  • Stereoisomerism

Substances

  • Biological Products
  • Epoxy Compounds
  • Ethers
  • Furans
  • tetrahydrofuran
  • Bromine