The Krüppel-like zinc finger protein Glis2 functions as a negative modulator of the Wnt/beta-catenin signaling pathway

FEBS Lett. 2007 Mar 6;581(5):858-64. doi: 10.1016/j.febslet.2007.01.058. Epub 2007 Feb 2.

Abstract

To gain insight into the mechanism by which Gli-similar 2 (Glis2) regulates transcription, we performed yeast-two hybrid cDNA library screening using Glis2 as bait. This screening identified beta-catenin as a potential Glis2-interacting protein. Mammalian two-hybrid, co-immunoprecipitation, and GST-pulldown analyses supported the interaction between Glis2 and beta-catenin. Pulldown analyses with several Glis2 deletion mutants indicated that the 1st zinc finger motif of Glis2 is critical for its interaction with beta-catenin, while the armadillo repeats of beta-catenin are important in its interaction with Glis2. Reporter analyses showed that Glis2 represses T-cell factor (TCF)-mediated transcriptional activation. In addition, Glis2 represses the expression of the TCF target gene cyclin D1. Our results indicate that Glis2 interacts with beta-catenin and suggest that Glis2 functions as a negative modulator of beta-catenin/TCF-mediated transcription.

Publication types

  • Research Support, N.I.H., Intramural

MeSH terms

  • Cell Line
  • Cell Nucleus / metabolism
  • Cyclin D
  • Cyclins / genetics
  • Humans
  • In Vitro Techniques
  • Kruppel-Like Transcription Factors / chemistry
  • Kruppel-Like Transcription Factors / genetics
  • Kruppel-Like Transcription Factors / metabolism*
  • Promoter Regions, Genetic
  • Protein Binding
  • Recombinant Proteins / chemistry
  • Recombinant Proteins / genetics
  • Recombinant Proteins / metabolism
  • Sequence Deletion
  • Signal Transduction
  • TCF Transcription Factors / metabolism
  • Transcriptional Activation
  • Two-Hybrid System Techniques
  • Wnt Proteins / genetics
  • Wnt Proteins / metabolism*
  • Zinc Fingers
  • beta Catenin / chemistry
  • beta Catenin / genetics
  • beta Catenin / metabolism*

Substances

  • CTNNB1 protein, human
  • Cyclin D
  • Cyclins
  • GLIS2 protein, human
  • Kruppel-Like Transcription Factors
  • Recombinant Proteins
  • TCF Transcription Factors
  • Wnt Proteins
  • beta Catenin