Effects of milnacipran and fluvoxamine on hyperemotional behaviors and the loss of tryptophan hydroxylase-positive cells in olfactory bulbectomized rats

Psychopharmacology (Berl). 2007 May;191(4):857-65. doi: 10.1007/s00213-007-0699-x. Epub 2007 Feb 22.

Abstract

Rationale: It has been reported that many of the behavioral and serotonergic neuronal changes observed in olfactory bulbectomy (OBX) were improved by subchronic administration of a variety of antidepressants.

Objective: We examined the effects of subchronic treatment with milnacipran, a dual serotonin and noradrenaline reuptake inhibitors (SNRIs) and fluvoxamine, selective serotonin reuptake inhibitors (SSRI) in the OBX-induced hyperemotional behaviors and tryptophan hydroxylase (TPH), rate-limiting enzyme of 5-HT.

Materials and methods: The olfactory bulbs were removed by suction. Drugs were administered p.o. once daily for 8 days beginning 14 days post-surgery. The hyperemotionality behaviors of OBX rats were measured by rating scale and in the elevated plus-maze test.

Results: OBX rats, after milnacipran or fluvoxamine treatment, showed significant decrease in the score of hyperemotional responses on 7th day as compared with vehicle-treated OBX rats. In addition, milnacipran and fluvoxamine in OBX rats respectively produced a significant increase in the percentage of time spent in and number of entries into open arms in the elevated plus maze test. Furthermore, when 5-HTnergic neuronal function was examined using antibodies against tryptophan hydroxylase (TPH) following the behavioral tests, fluvoxamine significantly reversed the loss of TPH-positive cells produced by OBX in the dorsal raphe.

Conclusion: We demonstrated that chronic treatment with milnacipran or fluvoxamine was effective to improve both the hyperemotional behavior and the loss of TPH-positive cells seen in OBX rats.

MeSH terms

  • Adrenergic Uptake Inhibitors / pharmacology*
  • Animals
  • Behavior, Animal / drug effects*
  • Cyclopropanes / pharmacology*
  • Dose-Response Relationship, Drug
  • Emotions / drug effects*
  • Fluvoxamine / pharmacology*
  • Male
  • Milnacipran
  • Motor Activity / drug effects
  • Neurons / drug effects
  • Neurons / enzymology
  • Olfactory Bulb / surgery
  • Raphe Nuclei / cytology
  • Raphe Nuclei / drug effects*
  • Raphe Nuclei / enzymology
  • Rats
  • Rats, Wistar
  • Selective Serotonin Reuptake Inhibitors / pharmacology*
  • Serotonin / metabolism
  • Time Factors
  • Tryptophan Hydroxylase / metabolism*

Substances

  • Adrenergic Uptake Inhibitors
  • Cyclopropanes
  • Serotonin Uptake Inhibitors
  • Serotonin
  • Tryptophan Hydroxylase
  • Milnacipran
  • Fluvoxamine