The effect of the controlled release of basic fibroblast growth factor from ionic gelatin-based hydrogels on angiogenesis in a murine critical limb ischemic model

Biomaterials. 2007 Jun;28(16):2646-54. doi: 10.1016/j.biomaterials.2007.01.044. Epub 2007 Feb 12.

Abstract

The localized delivery of exogenous, angiogenic growth factors has become a promising alternative treatment of peripheral artery disease (PAD) and critical limb ischemia. In the present study, we describe the development of a novel controlled release vehicle to promote angiogenesis in a murine critical limb ischemic model. Ionic, gelatin-based hydrogels were prepared by the carbodiimide-mediated amidation reaction between the carboxyl groups of gelatin or poly-L-glutamic acid molecules and the amine groups of poly-L-lysine or gelatin molecules, respectively. The degree of swelling of the synthesized hydrogels was assessed as a function of EDC/NHS ratios and the pH of the equilibrating medium, while the release kinetic profile of basic fibroblast growth factor (FGF-2) was evaluated in human fibroblast cultures. The degree of swelling (DS) decreased from 26.5+/-1.7 to 18.5+/-2.4 as the EDC concentration varied from 0.75 to 2.5 mg/ml. Eighty percent of the FGF-2 was released at controlled rates from gelatin-polylysine (gelatin-PLL) and gelatin-polyglutamic acid (gelatin-PLG) hydrogel scaffolds over a period of 28 days. Cell adhesion studies revealed that the negatively charged surface of the gelatin-PLG hydrogels exhibited superior adhesion capabilities in comparison to gelatin-PLL and control gelatin surfaces. Laser Doppler perfusion imaging as well as CD31(+) capillary immunostaining demonstrated that the controlled release of FGF-2 from ionic gelatin-based hydrogels is superior in promoting angiogenesis in comparison to the bolus administration of the growth factor. Over 4 weeks, FGF-2 releasing gelatin-PLG hydrogels exhibited marked reperfusion with a Doppler ratio of 0.889 (+/-0.04) which was 69.3% higher than in the control groups.

Publication types

  • Evaluation Study
  • Research Support, N.I.H., Extramural

MeSH terms

  • Animals
  • Biocompatible Materials / chemistry
  • Biocompatible Materials / metabolism
  • Cell Adhesion / physiology
  • Cells, Cultured
  • Delayed-Action Preparations
  • Drug Carriers* / chemistry
  • Drug Carriers* / metabolism
  • Extremities / blood supply
  • Extremities / pathology
  • Fibroblast Growth Factor 2 / metabolism*
  • Gelatin / chemistry*
  • Gelatin / metabolism
  • Humans
  • Hydrogels / chemistry*
  • Ischemia / drug therapy
  • Laser-Doppler Flowmetry
  • Mice
  • Mice, Inbred BALB C
  • Molecular Structure
  • Neovascularization, Physiologic*

Substances

  • Biocompatible Materials
  • Delayed-Action Preparations
  • Drug Carriers
  • Hydrogels
  • Fibroblast Growth Factor 2
  • Gelatin