In vitro and in vivo antiallergic effects of Glycyrrhiza glabra and its components

Planta Med. 2007 Mar;73(3):257-61. doi: 10.1055/s-2007-967126. Epub 2007 Feb 28.

Abstract

Licorice (Glycyrrhiza glabra L., Leguminosae) is frequently used in traditional medicine to treat inflammatory and allergic diseases. In this study, the main components (glycyrrhizin, 18beta-glycyrrhetinic acid, isoliquiritin, and liquiritigenin) were isolated from licorice, and their anti-allergic effects, such as antiscratching behavior and IgE production-inhibitory activity, were evaluated both in vitro and in vivo. Liquiritigenin and 18beta-glycyrrhetinic acid most potently inhibited the degranulation of RBL-2H3 cells induced by IgE with the antigen (DNP-HSA) and rat peritoneal mast cells induced by compound 48/80. Liquiritigenin and 18beta-glycyrrhetinic acid potently inhibited the passive cutaneous anaphylactic reaction as well as the scratching behavior in mice induced by compound 48/80. These components inhibited the production of IgE in ovalbumin-induced asthma mice but liquiritigenin had little effect. This suggests that the antiallergic effects of licorice are mainly due to glycyrrhizin, 18beta-glycyrrhetinic acid, and liquiritigenin, which can relieve IgE-induced allergic diseases such as dermatitis and asthma.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Anti-Allergic Agents / administration & dosage
  • Anti-Allergic Agents / chemistry
  • Anti-Allergic Agents / pharmacology*
  • Anti-Allergic Agents / therapeutic use
  • Asthma / chemically induced
  • Asthma / prevention & control*
  • Behavior, Animal / drug effects
  • Glycyrrhiza*
  • Immunoglobulin E / metabolism
  • Male
  • Mice
  • Mice, Inbred BALB C
  • Mice, Inbred ICR
  • Ovalbumin
  • Passive Cutaneous Anaphylaxis
  • Phytotherapy*
  • Plant Extracts / administration & dosage
  • Plant Extracts / chemistry
  • Plant Extracts / pharmacology*
  • Plant Extracts / therapeutic use
  • Plant Roots
  • p-Methoxy-N-methylphenethylamine

Substances

  • Anti-Allergic Agents
  • Plant Extracts
  • Immunoglobulin E
  • p-Methoxy-N-methylphenethylamine
  • Ovalbumin