PACAP type I receptor transactivation is essential for IGF-1 receptor signalling and antiapoptotic activity in neurons

EMBO J. 2007 Mar 21;26(6):1542-51. doi: 10.1038/sj.emboj.7601608. Epub 2007 Mar 1.

Abstract

Insulin-like growth factor-1 (IGF-1) and pituitary adenylyl cyclase activating polypeptide (PACAP) are both potent neurotrophic and antiapoptotic factors, which exert their effects via phosphorylation cascades initiated by tyrosine kinase and G-protein-coupled receptors, respectively. Here, we have adapted a recently described phosphoproteomic approach to neuronal cultures to characterize the phosphoproteomes generated by these neurotrophic factors. Unexpectedly, IGF-1 and PACAP increased the phosphorylation state of a common set of proteins in neurons. Using PACAP type 1 receptor (PAC1R) null mice, we showed that IGF-1 transactivated PAC1Rs constitutively associated with IGF-1 receptors. This effect was mediated by Src family kinases, which induced PAC1R phosphorylation on tyrosine residues. PAC1R transactivation was responsible for a large fraction of the IGF-1-associated phosphoproteome and played a critical role in the antiapoptotic activity of IGF-1. Hence, in contrast to the general opinion that the trophic activity of IGF-1 is solely mediated by tyrosine kinase receptor-associated signalling, we show that it involves a more complex signalling network dependent on the PAC1 Gs-protein-coupled receptor in neurons.

Publication types

  • Comparative Study
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Animals
  • Apoptosis / physiology*
  • Cyclic AMP / metabolism
  • Electrophoresis, Gel, Two-Dimensional
  • Immunoblotting
  • Immunohistochemistry
  • Immunoprecipitation
  • Insulin-Like Growth Factor I / metabolism*
  • Iodine Radioisotopes / metabolism
  • Mice
  • Mice, Inbred C57BL
  • Neurons / metabolism
  • Neurons / physiology*
  • Phosphoproteins / metabolism
  • Phosphorylation
  • Receptors, Pituitary Adenylate Cyclase-Activating Polypeptide, Type I / metabolism*
  • Signal Transduction / physiology*
  • Spectrometry, Mass, Matrix-Assisted Laser Desorption-Ionization
  • Transcriptional Activation / physiology*

Substances

  • Iodine Radioisotopes
  • Phosphoproteins
  • Receptors, Pituitary Adenylate Cyclase-Activating Polypeptide, Type I
  • Insulin-Like Growth Factor I
  • Cyclic AMP