A novel corepressor, BCoR-L1, represses transcription through an interaction with CtBP

J Biol Chem. 2007 May 18;282(20):15248-57. doi: 10.1074/jbc.M700246200. Epub 2007 Mar 22.

Abstract

Corepressors play a crucial role in negative gene regulation and are defective in several diseases. BCoR is a corepressor for the BCL6 repressor protein. Here we describe and functionally characterize BCoR-L1, a homolog of BCoR. When tethered to a heterologous promoter, BCoR-L1 is capable of strong repression. Like other corepressors, BCoR-L1 associates with histone deacetylase (HDAC) activity. Specifically, BCoR-L1 coprecipitates with the Class II HDACs, HDAC4, HDAC5, and HDAC7, suggesting that they are involved in its role as a transcriptional repressor. BCoR-L1 also interacts with the CtBP corepressor through a CtBP-interacting motif in its amino terminus. Abrogation of the CtBP binding site within BCoR-L1 partially relieves BCoR-L1-mediated transcriptional repression. Furthermore, BCoR-L1 is located on the E-cadherin promoter, a known CtBP-regulated promoter, and represses the E-cadherin promoter activity in a reporter assay. The inhibition of BCoR-L1 expression by RNA-mediated interference results in derepression of E-cadherin in cells that do not normally express E-cadherin, indicating that BCoR-L1 contributes to the repression of an authentic endogenous CtBP target.

Publication types

  • Research Support, Non-U.S. Gov't

MeSH terms

  • Alcohol Oxidoreductases / genetics
  • Alcohol Oxidoreductases / metabolism*
  • Amino Acid Motifs / genetics
  • Animals
  • Binding Sites / genetics
  • Cadherins / biosynthesis
  • Cadherins / genetics
  • Cell Line
  • DNA-Binding Proteins / genetics
  • DNA-Binding Proteins / metabolism*
  • Gene Expression Regulation / physiology*
  • Histone Deacetylases / genetics
  • Histone Deacetylases / metabolism
  • Humans
  • Mice
  • Multiprotein Complexes / genetics
  • Multiprotein Complexes / metabolism
  • Promoter Regions, Genetic / physiology
  • Protein Binding / genetics
  • Proto-Oncogene Proteins c-bcl-6
  • RNA Interference
  • Repressor Proteins / genetics
  • Repressor Proteins / metabolism*

Substances

  • BCL6 protein, human
  • BCORL1 protein, human
  • Bcl6 protein, mouse
  • Cadherins
  • DNA-Binding Proteins
  • Multiprotein Complexes
  • Proto-Oncogene Proteins c-bcl-6
  • Repressor Proteins
  • Alcohol Oxidoreductases
  • C-terminal binding protein
  • Histone Deacetylases