JB6 murine epidermal cell lines sensitive and resistant to 12-O-tetradecanoylphorbol-13-acetate (TPA)-induced transformation exhibit differential arachidonic acid metabolism in response to TPA and the calcium ionophore A23187

Carcinogenesis. 1992 Feb;13(2):189-92. doi: 10.1093/carcin/13.2.189.

Abstract

In a study of arachidonic acid metabolism in murine epidermal JB6 cells, promoter-sensitive (P+) and promoter-resistant (P-) variants, labeled with [3H]arachidonic acid, were treated successively with 12-O-tetradecanoylphorbol-13-acetate (TPA) and the calcium ionophore A23187. Released radiolabel was separated by HPLC and identified by coelution of standards. Prostacyclin release was then quantified by radioimmunoassay for 6-keto prostaglandin (PG)F1 alpha. A23187 alone resulted in a small but significant enhanced release of radiolabel from both cell variants (0.7 +/- 0.2% for P- and 0.6 +/- 0.3% for P+ cells; mean +/- SD). Treatment with TPA and subsequent treatment with A23187 resulted in a synergistically enhanced release of radiolabel from both cell variants (4.1 +/- 0.8% for P- and 3.4 +/- 0.9% for P+ cells) relative to that with either agent alone. Although the predominant product for each treatment regimen was prostaglandin E2 (PGE2), the TPA-resistant cells (P-) released significantly more 6-keto PGF1 alpha, a stable breakdown product of PGI2, than did the TPA-sensitive (P+) cells. These results indicate differential arachidonic acid metabolism between JB6 cell variants resistant and sensitive to TPA-induced transformation.

Publication types

  • Comparative Study
  • Research Support, U.S. Gov't, P.H.S.

MeSH terms

  • 6-Ketoprostaglandin F1 alpha / metabolism*
  • Animals
  • Calcimycin / pharmacology*
  • Cell Line
  • Cell Line, Transformed / drug effects
  • Chromatography, High Pressure Liquid
  • Dinoprostone / metabolism*
  • Drug Resistance
  • Epoprostenol / analysis
  • Mice
  • Mice, Inbred BALB C
  • Radioimmunoassay
  • Skin / cytology
  • Skin / drug effects
  • Skin / metabolism*
  • Tetradecanoylphorbol Acetate / pharmacology*

Substances

  • Calcimycin
  • 6-Ketoprostaglandin F1 alpha
  • Epoprostenol
  • Dinoprostone
  • Tetradecanoylphorbol Acetate